Pascal and Francis Bibliographic Databases

Help

Search results

Your search

cc.\*:("002B02B09A")

Filter

A-Z Z-A Frequency ↓ Frequency ↑
Export in CSV

Document Type [dt]

A-Z Z-A Frequency ↓ Frequency ↑
Export in CSV

Publication Year[py]

A-Z Z-A Frequency ↓ Frequency ↑
Export in CSV

Discipline (document) [di]

A-Z Z-A Frequency ↓ Frequency ↑
Export in CSV

Language

A-Z Z-A Frequency ↓ Frequency ↑
Export in CSV

Author Country

A-Z Z-A Frequency ↓ Frequency ↑
Export in CSV

Results 1 to 25 of 4355

  • Page / 175
Export

Selection :

  • and

Role of dexmedetomidine in adults in the intensive care unit: An updateREARDON, David P; ANGER, Kevin E; ADAMS, Christopher D et al.American journal of health-system pharmacy. 2013, Vol 70, Num 9, pp 767-777, issn 1079-2082, 11 p.Article

Design, synthesis, and pharmacological evaluation of novel tetrahydroprotoberberine derivatives: Selective inhibitors of dopamine D1 receptorWANGKE QIAN; WEIJIAN LU; XUECHU ZHEN et al.Bioorganic & medicinal chemistry. 2012, Vol 20, Num 15, pp 4862-4871, issn 0968-0896, 10 p.Article

Quinoline- and isoquinoline-sulfonamide derivatives of LCAP as potent CNS multi-receptor-5-HT1A/5-HT2A/5-HT7 and D2/D3/D4-agents: The synthesis and pharmacological evaluationZAJDEL, Paweł; MARCINIEC, Krzysztof; PAWLOWSKI, Maciej et al.Bioorganic & medicinal chemistry. 2012, Vol 20, Num 4, pp 1545-1556, issn 0968-0896, 12 p.Article

Further SAR study on 11-O-substituted aporphine analogues: Identification of highly potent dopamine D3 receptor ligandsNA YE; QIANQIAN WU; LIYUAN ZHU et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 6, pp 1999-2008, issn 0968-0896, 10 p.Article

Assessment of dopamine D1 receptor affinity and efficacy of three tetracyclic conformationally-restricted analogs of SKF38393CLARK, Alia H; MCCORVY, John D; WATTS, Val J et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 18, pp 5420-5431, issn 0968-0896, 12 p.Article

Further structure―activity relationship studies on 8-substituted-3-[2-(diarylmethoxyethylidenyl)]-8-azabicyclo[3.2.1]octane derivatives at monoamine transportersCARARAS, Shaine A; IZENWASSER, Sari; WADE, Dean et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 24, pp 7551-7558, issn 0968-0896, 8 p.Article

Schizophrenia: A Systematic Review of the Disease State, Current Therapeutics and their Molecular Mechanisms of ActionSHIN, J. K; MALONE, D. T; CROSBY, I. T et al.Current medicinal chemistry. 2011, Vol 18, Num 9, pp 1380-1404, issn 0929-8673, 25 p.Article

Development of (S)-N6-2-(4-(Isoquinolin-1-yl)piperazin-1-yl)ethyl-N6-propyl-4,5,6, tetrahydrobenzo[d]-thiazole-2,6-diamine and Its Analogue as a D3 Receptor Preferring Agonist: potent in Vivo Activity in Parkinson's Disease Animal ModelsGHOST, Balaram; ANTONIO, Tamara; JUAN ZHEN et al.Journal of medicinal chemistry (Print). 2010, Vol 53, Num 3, pp 1023-1037, issn 0022-2623, 15 p.Article

Discovery of olodaterol, a novel inhaled β2-drenoceptor agonist with a 24 h bronchodilatory efficacyBOUYSSOU, Thierry; HOENKE, Christoph; KONETZKI, Ingo et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 4, pp 1410-1414, issn 0960-894X, 5 p.Article

Scope and Difficulty in Generating Theoretical Insights Regarding Ligand Recognition and Activation of the β2 Adrenergic ReceptorSORIANO-URSUA, Marvin A; TRUJILLO-FERRARA, José G; CORREA-BASURTO, José et al.Journal of medicinal chemistry (Print). 2010, Vol 53, Num 3, pp 923-932, issn 0022-2623, 10 p.Article

The identification of a selective dopamine D2 partial agonist, D3 antagonist displaying high levels of brain exposureHOLMES, Ian P; BLUNT, Richard J; HOWES, Claire M et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 6, pp 2013-2016, issn 0960-894X, 4 p.Article

1,3-Dioxolane-based ligands incorporating a lactam or imide moiety: Structure-affinity/activity relationship at α1-adrenoceptor subtypes and at 5-HT1A receptorsFRANCHINI, Silvia; PRANDI, Adolfo; CICHERO, Elena et al.European journal of medicinal chemistry. 2010, Vol 45, Num 9, pp 3740-3751, issn 0223-5234, 12 p.Article

Design, synthesis and in vitro evaluation of (R)-4-(2-(tert-butylamino)-1-hydroxyethyl)-2-(hydroxymethyl)phenyl hydrogen phenylboronate: A novel salbutamol derivative with high intrinsic efficacy on the β2 adrenoceptorSORIANO-URSUA, Marvin A; CORREA-BASURTO, José; VALENCIA-HERNANDEZ, Ignacio et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 19, pp 5623-5629, issn 0960-894X, 7 p.Article

Discovery and synthesis of novel luteolin derivatives as DAT agonistsJIANGEZHANG; XIANBOLIU; XINSHENGLEI et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 22, pp 7842-7848, issn 0968-0896, 7 p.Article

Novel imidazoline compounds as partial or full agonists of D2-like dopamine receptors inspired by I2-imidazoline binding sites ligand 2-BFIGIORGIONI, Gianfabio; AMBROSINI, Dario; CARRIERI, Antonio et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 19, pp 7085-7091, issn 0968-0896, 7 p.Article

Structure―activity relationships in 1,4-benzodioxan-related compounds. 10. Novel α1-adrenoreceptor antagonists related to openphendioxan: Synthesis, biological evaluation, and α1d computational studyCARRIERI, Antonio; PIERGENTILI, Alessandro; DEL BELLO, Fabio et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 19, pp 7065-7077, issn 0968-0896, 13 p.Article

Synthesis and structure-activity studies of benzyl ester meperidine and normeperidine derivatives as selective serotonin transporter ligandsXIAOBO GU; IZENWASSER, Sari; WADE, Dean et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 23, pp 8356-8364, issn 0968-0896, 9 p.Article

Synthesis and α1-adrenoceptor antagonist activity of tamsulosin analoguesSAGRATINI, Gianni; ANGELI, Piero; BUCCIONI, Michela et al.European journal of medicinal chemistry. 2010, Vol 45, Num 12, pp 5800-5807, issn 0223-5234, 8 p.Article

An Overview on Benzylisoquinoline Derivatives with Dopaminergic and Serotonergic ActivitiesCABEDO, N; BERENGUER, I; FIGADERE, B et al.Current medicinal chemistry. 2009, Vol 16, Num 19, pp 2441-2467, issn 0929-8673, 27 p.Article

Cell Membrane Chromatography Correlated with Functional Assay for Ligand-β-Adrenergic Receptor AffinitiesAIGUO ZENG; BINGXIANG YUAN; FAN ZHU et al.Chromatographia (Wiesbaden). 2009, Vol 69, Num 11-12, pp 1373-1377, issn 0009-5893, 5 p.Article

Discovery of a new series of monoamine reuptake inhibitors, the 1-amino-3-(1H-indol-1-yl)-3-phenylpropan-2-olsKIM, Callain Y; MAHANEY, Paige E; MCCONNELL, Oliver et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 17, pp 5029-5032, issn 0960-894X, 4 p.Article

Synthesis and Structure-Activity Relationships of Long-acting β2 Adrenergic Receptor Agonists Incorporating Arylsulfonamide GroupsPROCOPIOU, Panayiotis A; BARRETT, Victoria J; GUNTRIP, Stephen B et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 8, pp 2280-2288, issn 0022-2623, 9 p.Article

1,1'-Disubstituted Ferrocenes as Molecular Hinges in Mono- and Bivalent Dopamine Receptor Ligand!HUBER, Daniela; HUBNER, Harald; GMEINER, Peter et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 21, pp 6860-6870, issn 0022-2623, 11 p.Article

Structure-activity relationship of dopaminergic halogenated 1-benzyl-tetrahydroisoquinoline derivativesEL AOUAD, Noureddine; BERENGUER, Inmaculada; CABEDO, Nuria et al.European journal of medicinal chemistry. 2009, Vol 44, Num 11, pp 4616-4621, issn 0223-5234, 6 p.Article

Involvement of dopamine and opioids in the motivation to eat : influence of palatability, homeostatic state, and behavioral paradigmsFLAVIA BARBANO, M; LE SAUX, Maryvonne; CADOR, Martine et al.Psychopharmacologia. 2009, Vol 203, Num 3, pp 475-487, issn 0033-3158, 13 p.Article

  • Page / 175