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Ensemble of G Protein-Coupled Receptor Active States : Recent Achievements on G-Protein Coupled ReceptorsPARK, P. S.-H.Current medicinal chemistry. 2012, Vol 19, Num 8, pp 1146-1154, issn 0929-8673, 9 p.Article

A New Target for Diagnosis and Treatment of CNS Disorders: Agmatinergic SystemUZBAY, T.Current medicinal chemistry. 2012, Vol 19, Num 30, pp 5116-5121, issn 0929-8673, 6 p.Conference Paper

Decahydroquinoline amides as highly selective CB2 agonists: Role of selectivity on in vivo efficacy in a rodent model of analgesiaMANLEY, Peter J; ZARTMAN, Amy; YEH, Suzie et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 8, pp 2359-2364, issn 0960-894X, 6 p.Article

Design, synthesis and structure―activity relationships of (indo-3-yl) heterocyclic derivatives as agonists of the CB1 receptor. Discovery of a clinical candidateRATCLIFFE, Paul; ADAM, Julia M; EDWARDS, Darren et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 8, pp 2541-2546, issn 0960-894X, 6 p.Article

Histamine H3 Receptor (H3R) Antagonists and Inverse Agonists in the Treatment of Sleep Disorders : Advances in the pharmacological approach to sleep disordersBRODERICK, Meredith; MASRI, Tony.Current pharmaceutical design (Print). 2011, Vol 17, Num 15, pp 1426-1429, issn 1381-6128, 4 p.Article

Microwave-assisted synthesis of quinoline, isoquinoline, quinoxaline and quinazoline derivatives as CB2 receptor agonistsSAARI, Raimo; TÖRMÄ, Jonna-Carita; NEVALAINEN, Tapio et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 2, pp 939-950, issn 0968-0896, 12 p.Article

The synthesis and biological evaluation of 2-(3-methyl or 3-phenylisoxazol-5-yl)-3-aryl-8-thiabicyclo[3.2.1]octanesPURUSHOTHAM, Madhusudhan; SHERI, Anjaneyulu; PHAM-HUU, Duy-Phong et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 1, pp 48-51, issn 0960-894X, 4 p.Article

Triamino pyrimidines and pyridines as histamine H4 receptor modulatorsMEDUNA, Steven P; SAVALL, Brad M; HUI CAI et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 10, pp 3113-3116, issn 0960-894X, 4 p.Article

Aryl 1,4-diazepane compounds as potent and selective CB2 agonists: Optimization of drug-like properties and target independent parametersZINDELL, Renée; WALKER, Edward R; KAPLITA, Paul et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 14, pp 4276-4280, issn 0960-894X, 5 p.Article

Synthesis and pharmacological evaluation of indole-based sigma receptor ligandsMESANGEAU, Christophe; AMATA, Emanuele; ALSHARIF, Walid et al.European journal of medicinal chemistry. 2011, Vol 46, Num 10, pp 5154-5161, issn 0223-5234, 8 p.Article

Endocannabinoid system dysfunction in mood and related disordersASHTON, C. H; MOORE, P. B.Acta psychiatrica scandinavica. 2011, Vol 124, Num 4, pp 250-261, issn 0001-690X, 12 p.Article

Endogenous ligand for an orphan receptorWOLF, George.Nutrition reviews. 2010, Vol 68, Num 5, pp 316-318, issn 0029-6643, 3 p.Article

Sigma-1 ligands: Tic-hydantoin as a key pharmacophoreTOUSSAINT, Marion; MOUSSET, Deborah; FOULON, Catherine et al.European journal of medicinal chemistry. 2010, Vol 45, Num 1, pp 256-263, issn 0223-5234, 8 p.Article

Synthesis and characterization of N,N-dialkyl and N-alkyl-N-aralkyl fenpropimorph-derived compounds as high affinity ligands for sigma receptorsHAJIPOUR, Abdol R; FONTANILLA, Dominique; CHU, Uyen B et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 12, pp 4397-4404, issn 0968-0896, 8 p.Article

Synthesis and pharmacology of 1-methoxy analogs of CP-47,497HUFFMAN, John W; HEPBURN, Seon A; REGGIO, Patricia H et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 15, pp 5475-5482, issn 0968-0896, 8 p.Article

Synthesis and structure-activity relationship of 1,2,4-triazole-containing diarylpyrazolyl carboxamide as CB1 cannabinoid receptor-ligandHEE JEONG SEO; MIN JU KIM; SUK HO LEE et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 3, pp 1149-1162, issn 0968-0896, 14 p.Article

Discovery of substituted benzyl tetrazoles as histamine H3 receptor antagonistsDAVENPORT, Adam J; STIMSON, Christopher C; CORSI, Massimo et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 17, pp 5165-5169, issn 0960-894X, 5 p.Article

Investigation of 4-piperidinols as novel H3 antagonistsANDERSON, James T; CAMPBELL, Michael; JIANMIN WANG et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 21, pp 6246-6249, issn 0960-894X, 4 p.Article

Synthesis and biological evaluation of new N-alkyl 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides as cannabinoid receptor ligandsSILVESTRI, Romano; LIGRESTI, Alessia; CARAI, Mauro Antonio Maria et al.European journal of medicinal chemistry. 2010, Vol 45, Num 12, pp 5878-5886, issn 0223-5234, 9 p.Article

Cannabinoid CB2 Receptors in Health and DiseasePATEL, K. D; DAVISON, J. S; PITTMAN, Q. J et al.Current medicinal chemistry. 2010, Vol 17, Num 14, pp 1394-1410, issn 0929-8673, 17 p.Article

1,4-Diazepanes derived from (S)-serine : Homopiperazines with improved σ1 (sigma) receptor affinity and selectivityBEDÜRFTIG, Stephan; WÜNSCH, Bernhard.European journal of medicinal chemistry. 2009, Vol 44, Num 2, pp 519-525, issn 0223-5234, 7 p.Article

6-Methoxy-N-alkyl Isatin Acylhydrazone Derivatives as a Novel Series of Potent Selective Cannabinoid Receptor 2 Inverse Agonists : Design, Synthesis, and Binding Mode PredictionDIAZ, Philippe; PHATAK, Sharangdhar S; JIJUN XU et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 2, pp 433-444, issn 0022-2623, 12 p.Article

Bioisosteric replacement of the hydrazide pharmacophore of the cannabinoid-1 receptor antagonist SR141716A. Part I: Potent, orally-active 1,4-disubstituted imidazolesDOW, Robert L; HADCOCK, John R; SCOTT, Dennis O et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 18, pp 5351-5354, issn 0960-894X, 4 p.Article

Brain-penetrating 2-aminobenzimidazole H1-antihistamines for the treatment of insomniaCOON, Timothy; MOREE, Wilna J; WEN, Jenny et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 15, pp 4380-4384, issn 0960-894X, 5 p.Article

Design and synthesis of novel tri-aryl CB2 selective cannabinoid ligandsBHATTACHARJEE, Himanshu; GURLEY, Steven N; MOORE, Bob M et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 6, pp 1691-1693, issn 0960-894X, 3 p.Article

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