2-Alkenylthieno[2,3-b]pyridine-5-carbonitriles : Potent and selective inhibitors of PKCθTUMEY, L. Nathan; BOSCHELLI, Diane H; LEE, Julie et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 15, pp 4420-4423, issn 0960-894X, 4 p.Article

4-Anilino-7-pyridyl-3-quinolinecarbonitriles as Src kinase inhibitorsNAN ZHANG; BIQI WU; BOSCHELLI, Diane H et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 17, pp 5071-5074, issn 0960-894X, 4 p.Article

Synthesis and inhibition of Src kinase activity by 7-ethenyl and 7-ethynyl-4-anilino-3-quinolinecarbonitrilesBARRIOS SOSA, Ana Carolina; BOSCHELLI, Diane H; FEI YE et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 9, pp 2155-2158, issn 0960-894X, 4 p.Article

Inhibition of Src kinase activity by 4-anilino-5,10-dihydropyrimido[4,5-b]quinolinesBOSCHELLI, Diane H; POWELL, Dennis; GOLAS, Jennifer M et al.Bioorganic & medicinal chemistry letters (Print). 2003, Vol 13, Num 18, pp 2977-2980, issn 0960-894X, 4 p.Article

Synthesis and PFCθ inhibitory activity of a series of 5-vinyl phenyl sulfonamide-3-pyridinecarbonitrilesSHIM, Jaechul; EID, Clark; LEE, Julie et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 23, pp 6575-6577, issn 0960-894X, 3 p.Article

5-Vinyl-3-pyridinecarbonitrile inhibitors of PKCθ: Optimization of enzymatic and functional activityNATHAN TUMEY, L; BHAGIRATH, Niala; BRENNAN, Agnes et al.Bioorganic & medicinal chemistry. 2009, Vol 17, Num 23, pp 7933-7948, issn 0968-0896, 16 p.Article

Facile preparation of new 4-phenylamino-3-quinolinecarbonitrile Src kinase inhibitors via 7-fluoro intermediates : Identification of potent 7-amino analogsBOSCHELLI, Diane H; BIQI WU; FEI YE et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 1, pp 405-412, issn 0968-0896, 8 p.Article

Optimization of 5-phenyl-3-pyridinecarbonitriles as PKCθ inhibitorsBOSCHELLI, Diane H; WANG, Daniel; PRASHAD, Amar S et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 13, pp 3623-3626, issn 0960-894X, 4 p.Article

Synthesis and Src kinase inhibitory activity of a series of 4-phenylamino-3-quinolinecarbonitrilesBOSCHELLI, Diane H; WANG, Yanong D; BOSCHELLI, Frank et al.Journal of medicinal chemistry (Print). 2001, Vol 44, Num 5, pp 822-833, issn 0022-2623Article

Inhibitors of Src tyrosine kinase : The preparation and structure-activity relationship of 4-anilino-3-cyanoquinolines and 4-anilinoquinazolinesWANG, Yanong D; MILLER, Karen; BOSCHELLI, Diane H et al.Bioorganic & medicinal chemistry letters (Print). 2000, Vol 10, Num 21, pp 2477-2480, issn 0960-894XArticle

C-5 Substituted heteroaryl 3-pyridinecarbonitriles as PKCθ inhibitors: Part ISUBRATH, Joan; WANG, Daniel; BIQI WU et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 18, pp 5423-5425, issn 0960-894X, 3 p.Article

Inhibition of Src kinase activity by 4-anilino-7-thienyl-3-quinolinecarbonitrilesBOSCHELLI, Diane H; WANG, Daniel Y; FEI YE et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 15, pp 2011-2014, issn 0960-894XArticle

Optimization of 5-vinylaryl-3-pyridinecarbonitriles as PKCθ inhibitorsBOSCHELLI, Diane H; SUBRATH, Joan; XIN XU et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 6, pp 1965-1968, issn 0960-894X, 4 p.Article

Optimization of 7-alkene-3-quinolinecarbonitriles as Src kinase inhibitorsBOSCHELLI, Diane H; WANG, Daniel; YAN WANG et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 9, pp 2924-2927, issn 0960-894X, 4 p.Article

First generation 5-vinyl-3-pyridinecarbonitrile PKCθ inhibitorsCHUANSHENG NIU; BOSCHELLI, Diane H; XIAOKE YANG et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 20, pp 5829-5832, issn 0960-894X, 4 p.Article

Pyrido[2,3-d]pyrimidin-7-one inhibitors of cyclin-dependent kinasesBARVIAN, Mark; BOSCHELLI, Diane H; LA, Frances et al.Journal of medicinal chemistry (Print). 2000, Vol 43, Num 24, pp 4606-4616, issn 0022-2623Article

Lead identification to generate 3-cyanoquinoline inhibitors of insulin-like growth factor receptor (IGF-1R) for potential use in cancer treatmentMILLER, Lori M; MAYER, Scott C; HESS KENNY, Cynthia et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 1, pp 62-66, issn 0960-894X, 5 p.Article

SKI-606, a Src/Abl inhibitor with in vivo activity in colon tumor xenograft modelsGALAS, Jennifer M; LUCAS, Judy; FANGBIAO LI et al.Cancer research (Baltimore). 2005, Vol 65, Num 12, pp 5358-5364, issn 0008-5472, 7 p.Article

SKI-606, a 4-anilino-3-quinolinecarbonitrile dual inhibitor of Src and Abl kinases, is a potent antiproliferative agent against chronic myelogenous leukemia cells in culture and causes regression of K562 xenografts in nude miceGOLAS, Jennifer M; ARNDT, Kim; ETIENNE, Carlo et al.Cancer research (Baltimore). 2003, Vol 63, Num 2, pp 375-381, issn 0008-5472, 7 p.Article

Optimization of 4-phenylamino-3-quinolinecarbonitriles as potent inhibitors of Src kinase activityBOSCHELLI, Diane H; FEI YE; TISCHLER, Mark et al.Journal of medicinal chemistry (Print). 2001, Vol 44, Num 23, pp 3965-3977, issn 0022-2623Article