Application of a water-soluble pyridyl disulfide amine linker for use in Cu-free click bioconjugationTHOMAS, Joshua D; BURKE, Terrence R.Tetrahedron letters. 2011, Vol 52, Num 33, issn 0040-4039, 4237, 4316-4319 [5 p.]Article

Investigation of Unanticipated Alkylation at the N(π) Position of a Histidyl Residue Under Mitsunobu Conditions and Synthesis of Orthogonally Protected Histidine AnaloguesWENJIAN QIAN; FA LIU; BURKE, Terrence R et al.Journal of organic chemistry. 2011, Vol 76, Num 21, pp 8885-8890, issn 0022-3263, 6 p.Article

Design and synthesis of a β-amino phosphotyrosyl mimetic suitably protected for peptide synthesisKYEONG LEE; MANCHAO ZHANG; DAJUN YANG et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 23, pp 3399-3401, issn 0960-894X, 3 p.Article

Design and synthesis of photoactivatable aryl diketo acid-containing HIV-1 integrase inhibitors as potential affinity probesXUECHUN ZHANG; MARCHAND, Christophe; POMMIER, Yves et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 5, pp 1205-1207, issn 0960-894X, 3 p.Article

Non-proteinogenic amino acids in the pThr-2 position of a pentamer peptide that confer high binding affinity for the polo box domain (PBD) of polo-like kinase 1 (Plk1)QIAN, Wen-Jian; PARK, Jung-Eun; LEE, Kyung S et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 24, pp 7306-7308, issn 0960-894X, 3 p.Article

Development of a phosphatase-stable phosphotyrosyl mimetic suitably protected for the synthesis of high-affinity Grb2 SH2 domain-binding ligandsWEI, Chang-Qing; BIHUA LI; RIBO GUO et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 19, pp 2781-2784, issn 0960-894X, 4 p.Article

Preparation of orthogonally protected (2S,3R)-2-amino-3-methyl-4-phosphonobutyric acid (Pmab) as a phosphatase-stable phosphothreonine mimetic and its use in the synthesis of polo-box domain-binding peptidesFA LIU; PARK, Jung-Eun; LEE, Kyung S et al.Tetrahedron (Oxford. Print). 2009, Vol 65, Num 47, issn 0040-4020, 9647, 9673-9679 [8 p.]Article

Protected aminooxyprolines for expedited library synthesis : Application to Tsg101-directed proline-oxime containing peptidesFA LIU; STEPHEN, Andrew G; FISHER, Robert J et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 3, pp 1096-1101, issn 0960-894X, 6 p.Article

Enantioselective synthesis of N^α-Fmoc protected (2S, 3R)-3-phenylpipecolic acid. A constrained phenylalanine analogue suitably protected for solid-phase peptide synthesisLIU, Ding-Guo; YANG GAO; XIANGZHU WANG et al.Journal of organic chemistry. 2002, Vol 67, Num 5, pp 1448-1452, issn 0022-3263Article

Macrocyclization in the design of a conformationally constrained Grb2 SH2 domain inhibitorYANG GAO; VOIGT, Johannes; WU, Jane X et al.Bioorganic & medicinal chemistry letters (Print). 2001, Vol 11, Num 14, pp 1889-1892, issn 0960-894XArticle

Selectivity and Mechanism of Action of a Growth Factor Receptor-Bound Protein 2 Src Homology 2 Domain Binding AntagonistGIUBELLINO, Alessio; SHI, Zhen-Dan; BOTTARO, Donald P et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 23, pp 7459-7468, issn 0022-2623, 10 p.Article

Examination of acylated 4-aminopiperidine-4-carboxylic acid residues in the phosphotyrosyl+1 position of grb2 SH2 domain-binding tripeptidesKANG, Sang-Uk; WON JUN CHOI; OISHI, Shinya et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 8, pp 1978-1982, issn 0022-2623, 5 p.Article

6,7-Dihydroxy-1-oxoisoindoline-4-sulfonamide-containing HIV-1 integrase inhibitorsXUE ZHI ZHAO; MADDALI, Kasthuraiah; SMITH, Steven J et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 24, pp 7309-7313, issn 0960-894X, 5 p.Article

A rapid oxime linker-based library approach to identification of bivalent inhibitors of the Yersinia pestis protein-tyrosine phosphatase, YopHFA LIU; RAMIN MOLLAAGHABABA HALCAMI; DYAS, Beverly et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 9, pp 2813-2816, issn 0960-894X, 4 p.Article

Examination of halogen substituent effects on HIV-1 integrase inhibitors derived from 2,3-dihydro-6,7-dihydroxy-1H-isoindol-1-ones and 4,5-dihydroxy-1H-isoindole-1,3(2H)-dionesXUE ZHI ZHAO; MADDALI, Kasthuraiah; VU, B. Christie et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 10, pp 2714-2717, issn 0960-894X, 4 p.Article

Identification of Shc Src Homology 2 Domain-Binding Peptoid-Peptide HybridsWON JUN CHOI; KIM, Sung-Eun; BOTTARO, Donald P et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 6, pp 1612-1618, issn 0022-2623, 7 p.Article

15-Deoxy-Δ^12,14-prostaglandin j₂ inhibits transcriptional activity of estrogen receptor-α via covalent modification of DNA-binding domainKIM, Han-Jong; KIM, Joon-Young; ZHAOJING MENG et al.Cancer research (Baltimore). 2007, Vol 67, Num 6, pp 2595-2602, issn 0008-5472, 8 p.Article

Inhibition of tumor metastasis by a growth factor receptor bound protein 2 src homology 2 domain-binding antagonistGIUBEFLINO, Alessio; YANG GAO; LEE, Sunmin et al.Cancer research (Baltimore). 2007, Vol 67, Num 13, pp 6012-6016, issn 0008-5472, 5 p.Article

Azido-containing diketo acid derivatives inhibit human immunodeficiency virus type 1 integrase in vivo and influence the frequency of deletions at two-long-terminal-repeat-circle junctionsSVAROVSKAIA, Evguenia S; BARR, Rebekah; XUECHUN ZHANG et al.Journal of virology. 2004, Vol 78, Num 7, pp 3210-3222, issn 0022-538X, 13 p.Article

Acylsulfonamide-containing PTP1B inhibitors designed to mimic an enzyme-bound water of hydrationLIU, Ding-Guo; YANG GAO; VOIGT, Johannes H et al.Bioorganic & medicinal chemistry letters (Print). 2003, Vol 13, Num 18, pp 3005-3007, issn 0960-894X, 3 p.Article

Coumarin-Based Inhibitors of Human NAD(P)H:Quinone Oxidoreductase-1. Identification, Structure-Activity, Off-Target Effects and In Vitro Human Pancreatic Cancer ToxicityNOLAN, Karen A; HE ZHAO; FAULDER, Paul F et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 25, pp 6316-6325, issn 0022-2623, 10 p.Article

Synthesis of tripeptides as potent Yersinia protein tyrosine phosphatase inhibitorsLEE, Kyeong; BOOVANAHALLI, Shanthaveerappa K; JUNG JUN LEE et al.Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 18, pp 4037-4042, issn 0960-894X, 6 p.Article

Tripeptide inhibitors of Yersinia protein-tyrosine phosphataseKYEONG LEE; YANG GAO; YAO, Zhu-Jun et al.Bioorganic & medicinal chemistry letters (Print). 2003, Vol 13, Num 15, pp 2577-2581, issn 0960-894X, 5 p.Article

Inhibition of human immunodeficiency virus type 1 integration by diketo derivativesPLUYMERS, Wim; PAIS, Godwin; VAN MAELE, Bénédicte et al.Antimicrobial agents and chemotherapy. 2002, Vol 46, Num 10, pp 3292-3297, issn 0066-4804, 6 p.Article

Development of tricyclic hydroxy-1H-pyrrolopyridine-trione containing HIV-1 integrase inhibitorsXUE ZHI ZHAO; MADDAL, Kasthuraiah; METIFIOT, Mathieu et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 10, pp 2986-2990, issn 0960-894X, 5 p.Article