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QSAR studies for diarylpyrimidines against HIV-1 reverse transcriptase wild-type and mutant strainsLIANG, Yong-Hong; CHEN, Fen-Er.European journal of medicinal chemistry. 2009, Vol 44, Num 2, pp 625-631, issn 0223-5234, 7 p.Article

A Facile and Efficient Asymmetric Synthesis of FlorfenicolFENG LI; WANG, Zhong-Hua; LEI ZHAO et al.Synlett (Stuttgart). 2011, Num 19, pp 2883-2885, issn 0936-5214, 3 p.Article

Direct Bifunctional Squaramide-Catalyzed Asymmetric N-Nitroso Aldol Reaction of Tertiary β-Carbonyl EstersYANG, Hong-Jun; LE DAI; YANG, Shi-Qiong et al.Synlett (Stuttgart). 2012, Num 6, pp 948-950, issn 0936-5214, 3 p.Article

Synthesis and in vitro anti-HIV evaluation of a new series of 6-arylmethyl-substituted S-DABOs as potential non-nucleoside HIV-1 reverse transcriptase inhibitorsWANG, Yue-Ping; CHEN, Fen-Er; DE CLERCQ, Erik et al.European journal of medicinal chemistry. 2009, Vol 44, Num 3, pp 1016-1023, issn 0223-5234, 8 p.Article

Non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 11: Structural modulations of diaryltriazines with potent anti-HIV activityXIONG, Yuan-Zhen; CHEN, Fen-Er; BALZARINI, Jan et al.European journal of medicinal chemistry. 2008, Vol 43, Num 6, pp 1230-1236, issn 0223-5234, 7 p.Article

Synthesis and biological evaluation of novel 6-substituted 5-alkyl-2-(arylcarbonylmethylthio)pyrimidin-4(3H)-ones as potent non-nucleoside HIV-1 reverse transcriptase inhibitorsWANG, Yue-Ping; CHEN, Fen-Er; DE CLERCQ, Erik et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 7, pp 3887-3894, issn 0968-0896, 8 p.Article

Synthesis and anti-HIV-1 activity evaluation of 5-alkyl-2-alkylthio-6-(arylcarbonyl or α -cyanoarylmethyl ) -3,4 -dihydropyrimidin -4 (3H) -ones as novel non-nucleoside HIV-1 reverse transcriptase inhibitorsLEI JI; CHEN, Fen-Er; DE CLERCQ, Erik et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 8, pp 1778-1786, issn 0022-2623, 9 p.Article

Efficient Asymmetric Synthesis of (2R,3R)-3-{(1R)-1-[tert-Butyl(dimethyl)-siloxy]ethyl}-4-oxoazetidin-2-yl AcetateHUANG, Jian-Ping; LEI ZHAO; GU, Shuang-Xi et al.Synthesis (Stuttgart). 2011, Num 4, pp 555-562, issn 0039-7881, 8 p.Article

Structural modifications of quinolone-3-carboxylic acids with anti-HIV activityHE, Qiu-Qin; GU, Shuang-Xi; JIA LIU et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 16, pp 5039-5045, issn 0968-0896, 7 p.Article

Synthesis and biological evaluation of (±)-benzhydrol derivatives as potent non-nucleoside HIV-1 reverse transcriptase inhibitorsMA, Xiao-Dong; XUAN ZHANG; YANG, Shi-Qiong et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 16, pp 4704-4709, issn 0968-0896, 6 p.Article

Synthesis and structure-activity relationship of novel diarylpyrimidines with hydromethyl linker (CH(OH)-DAPYs) as HIV-1 NNRTIsGU, Shuang-Xi; HE, Qiu-Qin; YANG, Shi-Qiong et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 17, pp 5117-5124, issn 0968-0896, 8 p.Article

Synthesis, structure—activity relationships, and docking studies of N-phenylarylformamide derivatives (PAFAs) as non-nucleoside HIV reverse transcriptase inhibitorsMA, Xiao-Dong; HE, Qiu-Qin; XUAN ZHANG et al.European journal of medicinal chemistry. 2012, Vol 58, pp 504-512, issn 0223-5234, 9 p.Article

Synthesis and biological evaluation of naphthyl phenyl ethers (NPEs) as novel nonnucleoside HIV-1 reverse transcriptase inhibitorsGU, Shuang-Xi; XUAN ZHANG; HE, Qiu-Qin et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 14, pp 4220-4226, issn 0968-0896, 7 p.Article

Design, synthesis and biological evaluation of cycloalkyl arylpyrimidines (CAPYs) as HIV-1 NNRTIsGU, Shuang-Xi; YANG, Shi-Qiong; HE, Qiu-Qin et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 23, pp 7093-7099, issn 0968-0896, 7 p.Article

Synthesis and biological activity of naphthyl-substituted (B-ring) benzophenone derivatives as novel non-nucleoside HIV-1 reverse transcriptase inhibitorsMA, Xiao-Dong; XUAN ZHANG; DAI, Hui-Fang et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 15, pp 4601-4607, issn 0968-0896, 7 p.Article

Hybrid diarylbenzopyrimidine non-nucleoside reverse transcriptase inhibitors as promising new leads for improved anti-HIV-1 chemotherapyZENG, Zhao-Sen; HE, Qiu-Qin; LIANG, Yong-Hong et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 14, pp 5039-5047, issn 0968-0896, 9 p.Article

Synthesis and anti-HIV activity of 2-naphthyl substituted DAPY analogues as non-nucleoside reverse transcriptase inhibitorsLIANG, Yong-Hong; HE, Qiu-Qin; ZENG, Zhao-Sen et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 13, pp 4601-4605, issn 0968-0896, 5 p.Article

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