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Role of dexmedetomidine in adults in the intensive care unit: An updateREARDON, David P; ANGER, Kevin E; ADAMS, Christopher D et al.American journal of health-system pharmacy. 2013, Vol 70, Num 9, pp 767-777, issn 1079-2082, 11 p.Article

Design, synthesis, and pharmacological evaluation of novel tetrahydroprotoberberine derivatives: Selective inhibitors of dopamine D1 receptorWANGKE QIAN; WEIJIAN LU; XUECHU ZHEN et al.Bioorganic & medicinal chemistry. 2012, Vol 20, Num 15, pp 4862-4871, issn 0968-0896, 10 p.Article

Quinoline- and isoquinoline-sulfonamide derivatives of LCAP as potent CNS multi-receptor-5-HT1A/5-HT2A/5-HT7 and D2/D3/D4-agents: The synthesis and pharmacological evaluationZAJDEL, Paweł; MARCINIEC, Krzysztof; PAWLOWSKI, Maciej et al.Bioorganic & medicinal chemistry. 2012, Vol 20, Num 4, pp 1545-1556, issn 0968-0896, 12 p.Article

Assessment of dopamine D1 receptor affinity and efficacy of three tetracyclic conformationally-restricted analogs of SKF38393CLARK, Alia H; MCCORVY, John D; WATTS, Val J et al.Bioorganic & medicinal chemistry. 2011, Vol 19, Num 18, pp 5420-5431, issn 0968-0896, 12 p.Article

Scope and Difficulty in Generating Theoretical Insights Regarding Ligand Recognition and Activation of the β2 Adrenergic ReceptorSORIANO-URSUA, Marvin A; TRUJILLO-FERRARA, José G; CORREA-BASURTO, José et al.Journal of medicinal chemistry (Print). 2010, Vol 53, Num 3, pp 923-932, issn 0022-2623, 10 p.Article

The identification of a selective dopamine D2 partial agonist, D3 antagonist displaying high levels of brain exposureHOLMES, Ian P; BLUNT, Richard J; HOWES, Claire M et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 6, pp 2013-2016, issn 0960-894X, 4 p.Article

Discovery and synthesis of novel luteolin derivatives as DAT agonistsJIANGEZHANG; XIANBOLIU; XINSHENGLEI et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 22, pp 7842-7848, issn 0968-0896, 7 p.Article

Novel imidazoline compounds as partial or full agonists of D2-like dopamine receptors inspired by I2-imidazoline binding sites ligand 2-BFIGIORGIONI, Gianfabio; AMBROSINI, Dario; CARRIERI, Antonio et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 19, pp 7085-7091, issn 0968-0896, 7 p.Article

Synthesis and α1-adrenoceptor antagonist activity of tamsulosin analoguesSAGRATINI, Gianni; ANGELI, Piero; BUCCIONI, Michela et al.European journal of medicinal chemistry. 2010, Vol 45, Num 12, pp 5800-5807, issn 0223-5234, 8 p.Article

Cell Membrane Chromatography Correlated with Functional Assay for Ligand-β-Adrenergic Receptor AffinitiesAIGUO ZENG; BINGXIANG YUAN; FAN ZHU et al.Chromatographia (Wiesbaden). 2009, Vol 69, Num 11-12, pp 1373-1377, issn 0009-5893, 5 p.Article

Discovery of a new series of monoamine reuptake inhibitors, the 1-amino-3-(1H-indol-1-yl)-3-phenylpropan-2-olsKIM, Callain Y; MAHANEY, Paige E; MCCONNELL, Oliver et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 17, pp 5029-5032, issn 0960-894X, 4 p.Article

1,1'-Disubstituted Ferrocenes as Molecular Hinges in Mono- and Bivalent Dopamine Receptor Ligand!HUBER, Daniela; HUBNER, Harald; GMEINER, Peter et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 21, pp 6860-6870, issn 0022-2623, 11 p.Article

Structure-activity relationship of dopaminergic halogenated 1-benzyl-tetrahydroisoquinoline derivativesEL AOUAD, Noureddine; BERENGUER, Inmaculada; CABEDO, Nuria et al.European journal of medicinal chemistry. 2009, Vol 44, Num 11, pp 4616-4621, issn 0223-5234, 6 p.Article

Discovery of a Novel Series of Biphenyl Benzoic Acid Derivatives as Potent and Selective Human β3-Adrenergic Receptor Agonists with Good Oral Bioavailability. Part IIMANISHI, Masashi; TOMISHIMA, Yasuyo; YAMAMOTO, Takao et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 6, pp 1925-1944, issn 0022-2623, 20 p.Article

Novel synthesis and pharmacological evaluation as α2-adrenoceptor ligands of O-phenylisouronium saltsGOONAN, Aine; KAHVEDZIC, Amila; RODRIGUEZ, Fernando et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 17, pp 8210-8217, issn 0968-0896, 8 p.Article

Structure-activity relationships of chiral selective norepinephrine reuptake inhibitors (sNRI) with increased oxidative stabilityHUDSON, Sarah; KIANKARIMI, Mehrak; WEN, Jenny et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 16, pp 4491-4494, issn 0960-894X, 4 p.Article

Synthesis and structure-activity relationships of selective norepinephrine reuptake inhibitors (sNRI) with a heterocyclic ring constraintHUDSON, Sarah; KIANKARIMI, Mehrak; ECCLES, Wendy et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 16, pp 4495-4498, issn 0960-894X, 4 p.Article

Synthesis of 4,5,6,7-tetrahydrothieno[3,2-c]pyridines and comparison with their isosteric 1,2,3,4-tetrahydroisoquinolines as inhibitors of phenylethanolamine N-methyltransferaseGRUNEWALD, Gary L; SEIM, Mitchell R; BHAT, Seema R et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 1, pp 542-559, issn 0968-0896, 18 p.Article

Synthesis of 1-arylpiperazyl-2-phenylcyclopropanes designed as antidopaminergic agents : Cyclopropane-based conformationally restricted analogs of haloperidolYAMAGUCHI, Kazuya; KAZUTA, Yuji; HIRANO, Kazufumi et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 19, pp 8875-8881, issn 0968-0896, 7 p.Article

Les sympathomimétiques en bref = Sympathomimetics in shortLa Revue Prescrire. 2008, Vol 28, Num DEC, pp 282-283, issn 0247-7750, 2 p., SUPArticle

Novel chiral isoxazole derivatives : Synthesis and pharmacological characterization at human β-adrenergic receptor subtypesDALLANOCE, Clelia; FRIGERIO, Fabio; DE AMICI, Marco et al.Bioorganic & medicinal chemistry. 2007, Vol 15, Num 7, pp 2533-2543, issn 0968-0896, 11 p.Article

Comment la noradrénaline est-elle utilisée en réanimation ? Une étude de terrain = How is norepinephrine used in intensive care? A field studyBIAZEJEWSKI, Sylvie; RAYMOND, Nathalie; LAGNAOUI, Rajaa et al.Thérapie (Paris). 2007, Vol 62, Num 2, pp 143-149, issn 0040-5957, 7 p.Article

Click chemistry based solid phase supported synthesis of dopaminergic phenylacetylenesRODRIGUEZ LOAIZA, Pilar; LÖBER, Stefan; HÜBNER, Harald et al.Bioorganic & medicinal chemistry. 2007, Vol 15, Num 23, pp 7248-7257, issn 0968-0896, 10 p.Article

High dopamine transporter selectivity can be displayed by remarkably simple non-nitrogen containing inhibitorsBOYE, Soren V; ORTEGA-CABALLERO, Fernando; SINNING, Steffen et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 21, pp 6019-6025, issn 0960-894X, 7 p.Article

α2-Adrenoreceptors Profile Modulation. 3. (R ) -(+ ) -m -Nitrobiphenyline, a New Efficient and α2C-Subtype Selective AgonistCRASSOUS, Pierre-Antoine; CARDINALETTI, Claudia; QUAGLIA, Wilma et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 16, pp 3964-3968, issn 0022-2623, 5 p.Article

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