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kw.\*:("Cyclohexanecarboxamide dérivé")

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Conjugate of neamine and 2-deoxystreptamine mimic connected by an amide bondUDUMULA, Venkatareddy; CHITTAPRAGADA, Maruthi; MARBLE, Jorden B et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 16, pp 4713-4715, issn 0960-894X, 3 p.Article

Highly Potent, Orally Available Anti-inflammatory Broad-Spectrum Chemokine InhibitorsFOX, David J; RECKLESS, Jill; LINGARD, Hannah et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 11, pp 3591-3595, issn 0022-2623, 5 p.Article

Oral cholesteryl ester transfer protein (CETP) inhibitors : A potential new approach for treating coronary artery diseaseSIKORSKI, James A.Journal of medicinal chemistry (Print). 2006, Vol 49, Num 1, pp 1-22, issn 0022-2623, 22 p.Article

Discovery of thiophene-2-carboxylic acids as potent inhibitors of HCV NS5B polymerase and HCV subgenomic RNA replication. Part 2: Tertiary amidesCHAN, Laval; PEREIRA, Oswy; ROY, Caroline et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 3, pp 797-800, issn 0960-894X, 4 p.Article

Design and synthesis of a biotinylated probe of COX-2 inhibitor nimesulide analog JCC76BO ZHONG; LAMA, Rati; SMITH, Kerri M et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 18, pp 5324-5327, issn 0960-894X, 4 p.Article

3D-QSAR studies with the aid of molecular docking for a series of non-steroidal FXR agonistsTAO ZHANG; ZHOU, Jun-Hong; SHI, Liang-Wei et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 8, pp 2156-2160, issn 0960-894X, 5 p.Article

Bis(2-(acylamino)phenyl) disulfides, 2-(acylamino)benzenethiols, and S-(2-(acylamino)phenyl) alkanethioates as novel inhibitors of cholesteryl ester transfer proteinSHINKAI, Hisashi; MAEDA, Kimiya; YAMASAKI, Takahiro et al.Journal of medicinal chemistry (Print). 2000, Vol 43, Num 19, pp 3566-3572, issn 0022-2623Article

Quantification of Lipophilicity of 1,2,4-Triazoles Using Micellar ChromatographyJANICKA, Matgorzata; STEPNIK, Katarzyna; PACHUTA-STEC, Anna et al.Chromatographia (Wiesbaden). 2012, Vol 75, Num 9-10, pp 449-456, issn 0009-5893, 8 p.Article

Novel cyclohexyl-amides as potent antibacterials targeting bacterial type IIA topoisomerasesMILES, Timothy J; BARFOOT, Christopher; GWYNN, Michael N et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 24, pp 7483-7488, issn 0960-894X, 6 p.Article

Evaluation of a 3-amino-8-azabicyclo[3.2.1]octane replacement in the CCR5 antagonist maravirocLEMOINE, Rémy C; PETERSEN, Ann C; SETTI, Lina et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 5, pp 1674-1676, issn 0960-894X, 3 p.Article

Design of inhibitors of scytalone dehydratase: Probing interactions with an asparagine carboxamideBASARAB, Gregory S; JORDAN, Douglas B; GEHRET, Troy C et al.Bioorganic & medicinal chemistry. 2002, Vol 10, Num 12, pp 4143-4154, issn 0968-0896, 12 p.Article

Retention-property relationships of 1,2,4-triazoles by micellar and reversed-phase liquid chromatographyJANICKA, Małgorzata; PACHUTA-STEC, Anna.Journal of separation science (Print). 2014, Vol 37, Num 12, pp 1419-1428, issn 1615-9306, 10 p.Article

Selectively Targeting T-and B-Cell Lymphomas : A Benzothiazole Antagonist of α4β1 IntegrinCARPENTER, Richard D; ANDREI, Mirela; AINA, Olulanu H et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 1, pp 14-19, issn 0022-2623, 6 p.Article

Vibriobactin Antibodies: A Vaccine StrategyBERGERON, Raymond J; BHARTI, Neelam; SINGH, Shailendra et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 12, pp 3801-3813, issn 0022-2623, 13 p.Article

Side Chain Flexibilities in the Human Ether-a-go-go Related Gene Potassium Channel (hERG) Together with Matched-Pair Binding Studies Suggest a New Binding Mode for Channel BlockersZACHARIAE, Ulrich; GIORDANETTO, Fabrizio; LEACH, Andrew G et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 14, pp 4266-4276, issn 0022-2623, 11 p.Article

Itk kinase inhibitors : Initial efforts to improve the metabolical stability and the cell activity of the benzimidazole leadMORIARTY, Kevin J; WINTERS, Michael; FARRELL, Thomas M et al.Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 20, pp 5537-5540, issn 0960-894X, 4 p.Article

Design, synthesis, and progress toward optimization of potent small molecule antagonists of CC chemokine receptor 8 (CCR8)GHOSH, Shomir; ELDER, Amy; BING GUAN et al.Journal of medicinal chemistry (Print). 2006, Vol 49, Num 9, pp 2669-2672, issn 0022-2623, 4 p.Article

3,4-Disubstituted azetidinones as selective inhibitors of the cysteine protease cathepsin K. Exploring P2 elements for selectivitySETTI, Eduardo L; DAVIS, Dana; CHUNG, Tobee et al.Bioorganic & medicinal chemistry letters (Print). 2003, Vol 13, Num 12, pp 2051-2053, issn 0960-894X, 3 p.Article

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