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DIMAPRIT, S-3-(N,N-DIMETHYLAMINO) PROPYL ISOTHIOUREA. A HIGHLY SPECIFIC HISTAMINE H2-RECEPTOR AGONIST. II. STRUCTURE-ACTIVITY CONSIDERATIONS.DURANT GJ; GANELLIN CR; PARSONS ME et al.1977; AGENTS AND ACTIONS; SWITZ.; DA. 1977; VOL. 7; NO 1; PP. 39-43; BIBL. 16 REF.Article

ANALEPTIC EFFECT OF CENTRALLY ADMINISTERED HISTAMINE H2-RECEPTOR AGONIST DIMAPRIT BUT NOT IMPROMIDINE IN URETHANE-ANAESTHETIZED RATSPAAKKARI I; KARPPANEN H.1982; NEUROPHARMACOLOGY; ISSN 0028-3908; GBR; DA. 1982; VOL. 21; NO 2; PP. 171-178; BIBL. 21 REF.Article

GASTRIC AND CARDIAC H-2 RECEPTOR EFFECTS OF DIMAPRIT, AND N'(ME), 5(ME) HISTAMINE IN CONSCIOUS DOGSHIRSCHOWITZ B; RENTZ J; MOLINA E et al.1980; EUROP. J. PHARMACOL.; NLD; DA. 1980; VOL. 61; NO 4; PP. 355-361; BIBL. 37 REF.Article

CIMETIDINE FAILS TO BLOCK FUNCTIONAL ANTAGONISM OF CARBACHOL BY HISTAMINE IN RAT TRACHEAEYRE P; BESNER RN.1979; RES. COMMUNIC. CHEM. PATHOL. PHARMACOL.; USA; DA. 1979; VOL. 24; NO 3; PP. 457-464; BIBL. 17 REF.Article

Antiproliferative and depigmenting effects of the histamine (H2) agonist dimaprit and its derivatives on human melanoma cellsFECHNER, G. A; PARSONS, P. G; MCEWAN, M. T et al.Biochemical pharmacology. 1992, Vol 43, Num 10, pp 2083-2090, issn 0006-2952Article

THE INFLUENCE OF 4-METHYLHISTAMINE, AN AGONIST OF HISTAMINE H2 RECEPTORS ON BODY TEMPERATURE IN RATSPILC A; NOWAK JZ.1980; NEUROPHARMACOLOGY; GBR; DA. 1980; VOL. 19; NO 8; PP. 773-775; BIBL. 17 REF.Article

STIMULATION OF GASTRIC ACID SECRETION BY DIMAPRIT IN UNANESTHETIZED RATSPETERSEN H; GROSSMAN MJ.1978; AGENTS AND ACTIONS; CHE; DA. 1978; VOL. 8; NO 6; PP. 566-567; BIBL. 4 REF.Article

N-Methyldimaprit (SK&F92054). A chemical control for the histamine H2-receptor agonist dimapritBLAKEMORE, R. C; GANELLIN, C. R; LEIGH, B. K et al.Collection sécurité. 1986, Vol 19, Num 1-2, pp 18-25, issn 0538-4818Article

INVESTIGATION OF THE ROLE OF HISTAMINE H1-RECEPTORS IN THE CONTROL OF GASTRIC ACID SECRETION IN THE RAT.BUNCE KT; PARSONS ME.1978; J. PHARM. PHARMACOL.; G.B.; DA. 1978; VOL. 30; NO 4; PP. 247-249; BIBL. 14 REF.Article

STIMULATION OF CELL PROLIFERATION BY HISTAMINE H2 RECEPTORS IN DIMETHYLHYDRAZINE-INDUCED ADENOCARCINOMATA.TUTTON PJM; BARKLA DH.1978; CELL BIOL., INTERNATION. REP.; G.B.; DA. 1978; VOL. 2; NO 2; PP. 199-202; BIBL. 14 REF.Article

STUDIO DI SOSTANZE ANALOGHE AL DIMAPRIT SULLA SECREZIONE GASTRICA IN VITRO = ETUDE DE SUBSTANCES ANALOGUES AU DIMAPRIT: ACTION SUR LA SECRETION GASTRIQUE IN VITROMORINI G; PLAZZI PV; BORDI F et al.1980; BOLL. SOC. ITAL. BIOL. SPER.; ITA; DA. 1980; VOL. 56; NO 1; PP. 88-94; ABS. ENG; BIBL. 7 REF.Article

EFFECTS OF DIMAPRIT, PROSTACYCLIN, AND ACETYLCHOLINE ON RENAL BLOOD FLOW AND FUNCTIONPAWLIK WW; JACOBSON ED; BANKS RO et al.1980; PROC. SOC. EXPER. BIOL. MED.; USA; DA. 1980; VOL. 163; NO 3; PP. 344-349; BIBL. 17 REF.Article

SPECIFIC ACTIVATION OF CYCLIC AMP-DEPENDENT PROTEIN KINASE (S) BY H2 HISTAMINE AGONISTS IN ISOLATED GASTRIC MUCOSAL CELLS FROM GUINEA-PIGMANGEAT P; MARCHIS MOUREN G; CHERET AM et al.1980; BIOCHIM. BIOPHYS. ACTA; NLD; DA. 1980; VOL. 629; NO 3; PP. 604-608; BIBL. 20 REF.Article

DIMAPRIT-(S-(3-(N,N-DIMETHYLAMINO) PROPYL) ISOTHIOUREA) - A HIGHLY SPECIFIC HISTAMINE H2-RECEPTOR AGONIST. I. PHARMACOLOGY.PARSONS ME; OWEN DAA; GANELLIN CR et al.1977; AGENTS AND ACTIONS; SWITZ.; DA. 1977; VOL. 7; NO 1; PP. 31-37; BIBL. 20 REF.Article

HISTAMINE-INDUCED RISE IN CORE TEMPERATURE OF CHLORAL-ANESTHETIZED RATS: MEDIATION BY H2-RECEPTORS LOCATED IN THE PREOPTICUS AREA OF HYPOTHALAMUSCOLBOC O; PROTAIS P; COSTENTIN J et al.1982; NEUROPHARMACOLOGY; ISSN 0028-3908; GBR; DA. 1982; VOL. 21; NO 1; PP. 45-50; BIBL. 32 REF.Article

AN INHIBITORY EFFECT OF HISTAMINE ON THE RAT ANOCOCCYGEUS MUSCLEAYOTUNDE ORIOWO M.1982; J. PHARM. PHARMACOL.; ISSN 0022-3573; GBR; DA. 1982; VOL. 34; NO 3; PP. 207-208; BIBL. 12 REF.Article

HISTAMINE RECEPTORS IN THE GUINEA-PIG DUODENUMBERTACCINI G; ZAPPIA L.1981; J. PHARM. PHARMACOL.; ISSN 0022-3573; GBR; DA. 1981; VOL. 33; NO 9; PP. 590-593; BIBL. 19 REF.Article

NEW INHIBITORS OF HISTAMINE-N-METHYLTRANSFERASEBEAVEN MA; SHAFF RE.1979; BIOCHEM. PHARMACOL.; GBR; DA. 1979; VOL. 28; NO 2; PP. 183-188; BIBL. 41 REF.Article

RELAXANT EFFECTS OF SELECTED BRONCHODILATORS ON EQUINE PULMONARY VEIN AND TRACHEAL SMOOTH MUSCLEHANNA J; EYRE P.1980; LUNG; DEU; DA. 1980; VOL. 158; NO 1; PP. 33-40; BIBL. 14 REF.Article

SENSORY RESPONSES OF HUMAN SKIN TO SYNTHETIC HISTAMINE ANALOGUES AND HISTAMINEDAVIES MG; GREAVES MW.1980; BRIT. J. CLIN. PHARMACOL.; GBR; DA. 1980; VOL. 9; NO 5; PP. 461-465; BIBL. 7 REF.Article

INHIBITION OF HISTAMINE METHYLATION IN VIVO BY THE DIMAPRIT ANALOG, SKF COMPOUND 91488BEAVEN MA; SHAFF RE.1979; AGENTS AND ACTIONS; CHE; DA. 1979; VOL. 9; NO 5-6; PP. 455-460; BIBL. 37 REF.Article

EFFECT OF DIMAPRIT ON GASTRIC ACID SECRETION IN CONSCIOUS CATSCARTER DC; IMPICCIATORE M; GROSSMAN MI et al.1978; AGENTS AND ACTIONS; CHE; DA. 1978; VOL. 8; NO 5; PP. 453-457; BIBL. 10 REF.Article

Histamine receptors on rat ocular surfaceUMEMOTO, M; TANAKA, H; MIICHI, H et al.Ophthalmic research. 1987, Vol 19, Num 4, pp 200-204, issn 0030-3747Article

Histamine inhibits interleukin 1 production by lipopolysaccharide-stimulated human peripheral blood monocytesDOHLSTEN, M; KALLAND, T; SJÖGREN, H.-O et al.Scandinavian journal of immunology (Print). 1988, Vol 27, Num 5, pp 527-532, issn 0300-9475Article

Effects of dimaprit on growth and differentiation of human promyelocytic cell line, HL-60KALINYAK, K. A; SAWUTZ, D. G; LAMPKIN, B. C et al.Life sciences (1973). 1985, Vol 36, Num 20, pp 1909-1916, issn 0024-3205Article

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