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MECHANISM OF ACTION OF METHOTREXATE. IV. FREE INTRACELLULAR METHOTREXATE REQUIRED TO SUPRESS DIHYDROFOLATE REDUCTION TO TETRAHYDROFOLATE BY EHRLICH ASCITES TUMOR CELLS IN VITRO.WHITE JC; GOLDMAN ID.1976; MOLEC. PHARMACOL.; U.S.A.; DA. 1976; VOL. 12; NO 5; PP. 711-719; BIBL. 41 REF.Article

INHIBITION OF THE MEMBRANE TRANSPORT OF FOLATES BY ANIONS RETAINED IN UREMIA = INHIBITION DU TRANSPORT MEMBRANAIRE DES FOLATES PAR LES ANIONS RETENUS DANS L'UREMIEJENNETTE JC; GOLDMAN ID.1975; J. LAB. CLIN. MED.; U.S.A.; DA. 1975; VOL. 86; NO 5; PP. 834-843; BIBL. 19 REF.Article

THE RELATIONSHIP AMONG TRANSPORT, INTRACELLULAR BINDING, AND INHIBITION OF RNA SYNTHESIS BY ACTINOMYCIN D IN EHRLICH ASCITES TUMOR CELLS IN VITRO. = RELATION ENTRE LE TRANSPORT, LA FIXATION INTRACELLULAIRE ET L'INHIBITION DE LA SYNTHESE D'ARN PAR L'ACTINOMYCINE D DANS LES CELLULES DE LA TUMEUR ASCITIQUE D'EHRLICH IN VITROBOWEN D; GOLDMAN ID.1975; CANCER RES.; U.S.A.; DA. 1975; VOL. 35; NO 11; PP. 3054-3060; BIBL. 35 REF.Article

EFFLUX IN ISOLATED HEPATOCYTES AS A POSSIBLE CORRELATE OF SECRETION IN VIVO: INDUCED EXIT OF THE FOLIC ACID ANALOG METHOTREXATE, BY DIBUTYRYL CYCLIC AMP OR ISOBUTYL METHYL XANTHINEGEWIRTZ DA; RANDOLPH JK; GOLDMAN ID et al.1981; BIOCHEM. BIOPHYS. RES. COMMUN.; ISSN 0006-291X; USA; DA. 1981; VOL. 101; NO 2; PP. 366-374; BIBL. 32 REF.Article

POTENT BILE SALT AND ORGANIC ANION INHIBITION OF METHOTREXATE UPTAKE AND ACCUMULATION IN THE FRESHLY ISOLATED RAT HEPATOCYTEGEWIRTZ DA; RANDOLPH JK; GOLDMAN ID et al.1980; CANCER RES.; USA; DA. 1980; VOL. 40; NO 6; PP. 1852-1857; BIBL. 43 REF.Article

THE MECHANISM OF ACTION OF METHOTREXATE. III. REQUIREMENT OF FREE INTRACELLULAR METHOTREXATE FOR MAXIMAL SUPPRESSION OF (14C) FORMATE INCORPORATION INTO NUCLEIC ACIDS AND PROTEIN = MECANISME DE L'ACTION DU METHOTREXATE. III. NECESSITE DE METHOTREXATE INTRACELLULAIRE LIBRE POUR LA SUPPRESSION MAXIMALE DE L'INCORPORATION DE FORMATE 14C DANS LES ACIDES NUCLEIQUES ET LES PROTEINESWHITE JC; LOFTFIELD S; GOLDMAN ID et al.1975; MOLEC. PHARMACOL.; U.S.A.; DA. 1975; VOL. 11; NO 3; PP. 287-297; BIBL. 1P.Article

TENIPOSIDE (VM-26)- AND ETOPOSIDE (VP-16-213)-INDUCED AUGMENTATION OF METHOTREXATE TRANSPORT AND POLYGLUTAMYLATION IN EHRLICH ASCITES TUMOR CELLS IN VITROYALOWICH JC; FRY DW; GOLDMAN ID et al.1982; CANCER RES.; USA; DA. 1982; VOL. 42; NO 9; PP. 3648-3653; BIBL. 36 REF.Article

AUGMENTATION OF THE INTRACELLULAR LEVELS OF POLYGLUTAMYL DERIVATIVES OF METHOTREXATE BY VINCRISTINE AND PROBENECID IN EHRLICH ASCITES TUMOR CELLSFRY DW; YALOWICH JC; GOLDMAN ID et al.1982; CANCER RES.; ISSN 0008-5472; USA; DA. 1982; VOL. 42; NO 7; PP. 2532-2536; BIBL. 25 REF.Article

K+-INDUCED ALTERATIONS OF ENERGETICS AND EXCHANGE DIFFUSION IN THE CARRIER-MEDIATED TRANSPORT OF THE FOLIC ACID ANALOG METHOTREXATE IN EHRLICH ASCITES TUMOR CELLSFRY DW; CYBULSKI RL; GOLDMAN ID et al.1980; BIOCHIM. BIOPHYS. ACTA; ISSN 0006-3002; NLD; DA. 1980; VOL. 603; NO 1; PP. 157-170; BIBL. 33 REF.Article

A REDUCTION IN ENERGY-DEPENDENT AMINO ACID TRANSPORT BY MICROTUBULAR INHIBITORS IN EHRLICH ASCITES TUMOR CELLS.FYFE MJ; LOFTFIELD S; GOLDMAN ID et al.1975; J. CELL. PHYSIOL.; G.B.; DA. 1975; VOL. 86; NO 2; PP. 201-212; BIBL. 1 P.Article

ADENOSINE STIMULATION OF UPHILL ADENINE TRANSPORT IN L1210 LEUKEMIA CELLS: EVIDENCE FOR A NOVEL COUNTERTRANSPORT MECHANISMCYBULSKI RL; FRY DW; GOLDMAN ID et al.1981; J. BIOL. CHEM.; ISSN 0021-9258; USA; DA. 1981; VOL. 256; NO 9; PP. 4455-4459; BIBL. 27 REF.Article

ALTERATIONS OF THE CARRIER-MEDIATED TRANSPORT OF AN ANIONIC SOLUTE, METHOTREXATE, BY CHARGED LIPOSOMES IN EHRLICH ASCITES TUMOR CELLSFRY DW; WHITE JC; GOLDMAN ID et al.1979; J. MEMBRANE BIOL.; USA; DA. 1979; VOL. 50; NO 2; PP. 123-140; BIBL. 49 REF.Article

A BASIS FOR FLUOROPYRIMIDINE-INDUCED ANTAGONISM TO METHOTREXATE IN EHRLICH ASCITES TUMOR CELLS IN VITRO.BOWEN D; WHITE JC; GOLDMAN ID et al.1978; CANCER RES.; U.S.A.; DA. 1978; VOL. 38; NO 1; PP. 219-222; BIBL. 31 REF.Article

RAPID FORMATION OF POLY-GAMMA -GLUTAMYL DERIVATIVES OF METHOTREXATE AND THEIR ASSOCIATION WITH DIHYDROFOLATE REDUCTASE AS ASSESSED BY HIGH PRESSURE LIQUID CHROMATOGRAPHY IN THE EHRLICH ASCITES TUMOR CELL IN VITROFRY DW; YALOWICH JC; GOLDMAN ID et al.1982; J. BIOL. CHEM.; ISSN 0021-9258; USA; DA. 1982; VOL. 257; NO 4; PP. 1890-1896; BIBL. 31 REF.Article

EFFECTS OF 2,4-DINITROPHENOL AND OTHER METABOLIC INHIBITORS ON THE BIDIRECTIONAL CARRIER FLUXES, NET TRANSPORT AND INTRACELLULAR BINDING OF METHOTREXATE IN EHRLICH ASCITES TUMOR CELLSFRY DW; WHITE JC; GOLDMAN ID et al.1980; CANCER RES.; ISSN 0008-5472; USA; DA. 1980; VOL. 40; NO 10; PP. 3669-3673; BIBL. 25 REF.Article

LACK OF STEREOSPECIFICITY AT CARBON 6 OF METHYLTETRAHYDROFOLATE TRANSPORT OF EHRLICH ASCITES TUMOR CELLS. CARRIER-MEDIATED TRANSPORT OF BOTH STEREOISOMERS.WHITE JC; BAILEY BD; GOLDMAN ID et al.1978; J. BIOL. CHEM.; U.S.A.; DA. 1978; VOL. 253; NO 1; PP. 242-245; BIBL. 29 REF.Article

ANALYSIS OF THE ROLE OF MEMBRANE TRANSPORT AND POLYGLUTAMATION OF METHOTREXATE IN GUT AND THE EHRLICH TUMOR IN VIVO AS FACTORS IN DRUG SENSITIVITY AND SELECTIVITY = ANALYSE DU ROLE DU TRANSPORT MEMBRANAIRE, DE LA POLYGLUTAMATION DU METHOTREXATE DANS LES INTESTINS ET LA TUMEUR D'EHRLICH IN VIVO COMME FACTEURS DE LA SENSIBILITE ET SELECTIVITE DE LA DROGUEFRY DW; ANDERSON LA; BORST M et al.1983; CANCER RESEARCH; ISSN 0008-5472; USA; DA. 1983; VOL. 43; NO 3; PP. 1087-1092; ABS. ENG; BIBL. 39 REF.; GRAPHArticle

TRANSPORT, BINDING, AND POLYGLUTAMATION OF METHOTREXATE IN FRESHLY ISOLATED RAT HEPATOCYTESGEWIRTZ DA; WHITE JC; RANDOLPH JK et al.1980; CANCER RES.; USA; DA. 1980; VOL. 40; NO 3; PP. 573-578; BIBL. 37 REF.Article

FORMATION OF METHOTREXATE POLYGLUTAMATES IN RAT HEPATOCYTESGEWIRTZ DA; WHITE JC; RANDOLPH JK et al.1979; CANCER RES.; USA; DA. 1979; VOL. 39; NO 8; PP. 2914-2918; BIBL. 37 REF.Article

RELATIONSHIP BETWEEN MEMBRANE TRANSPORT OF METHOTREXATE AND ENDOGENOUS CYCLIC ADENOSINE 3':5'-MONOPHOSPHATE IN THE EHRLICH ASCITES TUMORCOURTLAND WHITE J; CARCHMAN RA; FRY DW et al.1980; CANCER RES.; USA; DA. 1980; VOL. 40; NO 7; PP. 2400-2404; BIBL. 22 REF.Article

CHARACTERISTICS OF TRANSPORT OF 4-AMINO ANTIFOLATES AND FOLATE COMPOUNDS BY TWO LINES OF L 5178Y LYMPHOBLASTS, ONE WITH IMPAIRED TRANSPORT OF METHOTREXATEHILL BT; BAILEY BD; WHITE JC et al.1979; CANCER RES.; USA; DA. 1979; VOL. 39; NO 7 PART. 1; PP. 2440-2446; BIBL. 32 REF.Article

FOLYL AND ANTIFOLYL POLYGLUTAMATES. PROCEEDINGS OF A WORKSHOP HELD MAY 20-23, 1981, AT THE AIRLIE FOUNDATION, AIRLIE, VIRGINIAGOLDMAN ID ED; CHABNER BA ED; BERTINO JR ED et al.1983; ADVANCES IN EXPERIMENTAL MEDICINE AND BIOLOGY; ISSN 0065-2598; USA; DA. 1983; VOL. 163; X-425 P.; BIBL. DISSEM.Conference Paper

EXCHANGEABLE INTRACELLULAR METHOTREXATE LEVELS IN THE PRESENCE AND ABSENCE OF VINCRISTINE AT EXTRACELLULAR DRUG CONCENTRATIONS RELEVANT TO THOSE ACHIEVED IN HIGH-DOSE METHOTREXATE-FOLINIC ACID "RESCUE" PROTOCOLS. = TAUX DE METHOTREXATE INTRACELLULAIRE ECHANGEABLE EN LA PRESENCE ET EN L'ABSENCE DE VINCRISTINE AUX CONCENTRATIONS EXTRA CELLULAIRES DU MEDICAMENT EN RAPPORT AVEC CELLES OBTENUES DANS LES PROTOCOLES ASSOCIANT LE METHOTREXATE A DOSES ELEVEES ET L'ACIDE FOLINIQUE "ADJUVANT"GOLDMAN ID; VATSALA GUPTA; WHITE JC et al.1976; CANCER RES.; U.S.A.; DA. 1976; VOL. 36; NO 1; PP. 276-279; BIBL. 30 REF.Article

RAPID CATABOLISM OF 5-FLUOROURACIL IN FRESHLY ISOLATED RAT HEPATOCYTES AS ANALYZED BY HIGH PERFORMANCE LIQUID CHROMATOGRAPHYSOMMADOSSI JP; GEWIRTZ DA; DIASIO RB et al.1982; J. BIOL. CHEM.; ISSN 0021-9258; USA; DA. 1982; VOL. 257; NO 14; PP. 8171-8176; BIBL. 35 REF.Article

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