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Pharmacological characterization of the cannabinoid CB1 receptor PET ligand ortholog, [3H]MePPEPSUTER, Todd M; CHESTERFIELD, Amy K; CHUN BAO et al.European journal of pharmacology. 2010, Vol 649, Num 1-3, pp 44-50, issn 0014-2999, 7 p.Article

Pharmacological and behavioral properties of A-349821, a selective and potent human histamine H3 receptor antagonistESBENSHADE, Timothy A; FOX, Gerard B; FAGHIH, Ramin et al.Biochemical pharmacology. 2004, Vol 68, Num 5, pp 933-945, issn 0006-2952, 13 p.Article

Anxiogenic properties of an inverse agonist selective for α3 subunit-containing GABAA receptorsATACK, John R; HUTSON, Peter H; DAWSON, Gerard R et al.British journal of pharmacology. 2005, Vol 144, Num 3, pp 357-366, issn 0007-1188, 10 p.Article

ARB and Cardioprotection : NEW ASPECTS OF THE RENIN-ANGIOTENSIN ALDOSTERONE SYSTEM (RAAS) IN CARDIOVASCULAR DISEASEAKAZAWA, Hiroshi; YABUMOTO, Chizuru; YANO, Masamichi et al.Cardiovascular drugs and therapy. 2013, Vol 27, Num 2, pp 155-160, issn 0920-3206, 6 p.Article

Synthesis of constrained benzocinnolinone analogues of CEP-26401 (irdabisant) as potent, selective histamine H3 receptor inverse agonistsJOSEF, Kurt A; AIMONE, Lisa D; LYONS, Jacquelyn et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 12, pp 4198-4202, issn 0960-894X, 5 p.Article

Receptor-specific functional efficacies of alkyl imidazoles as dual histamine H3/H4 receptor ligandsKOTTKE, Tim; SANDER, Kerstin; WEIZEL, Lilia et al.European journal of pharmacology. 2011, Vol 654, Num 3, pp 200-208, issn 0014-2999, 9 p.Article

Molecular basis of melanocortin-4 receptor for AGRP inverse agonismMIN CHEN; CELIK, Ahmet; GEORGESON, Keith E et al.Regulatory peptides. 2006, Vol 136, Num 1-3, pp 40-49, issn 0167-0115, 10 p.Article

Some implications of receptor theory for in vivo assessment of agonists, antagonists and inverse agonistsNEGUS, S. Steuens.Biochemical pharmacology. 2006, Vol 71, Num 12, pp 1663-1670, issn 0006-2952, 8 p.Article

Involvement of cannabinoid CB2 receptor-mediated response and efficacy of cannabinoid CB2 receptor inverse agonist, JTE-907, in cutaneous inflammation in miceUEDA, Yoshifumi; MIYAGAWA, Naoki; MATSUI, Tomoko et al.European journal of pharmacology. 2005, Vol 520, Num 1-3, pp 164-171, issn 0014-2999, 8 p.Article

Interaction of valerian extracts of different polarity with adenosine receptors : Identification of isovaltrate as an inverse agonist at A1 receptorsLACHER, Svenja K; MAYER, Ralf; SICHARDT, Kathrin et al.Biochemical pharmacology. 2007, Vol 73, Num 2, pp 248-258, issn 0006-2952, 11 p.Article

SB265610 is an allosteric, inverse agonist at the human CXCR2 receptorBRADLEY, M. E; BOND, M. E; MANINI, J et al.British journal of pharmacology. 2009, Vol 158, Num 1, pp 328-338, issn 0007-1188, 11 p.Article

4,5-Dihydropyridazin-3-one derivatives as histamine H3 receptor inverse agonistsHUDKINS, Robert L; AIMONE, Lisa D; ZULLI, Allison L et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 194-198, issn 0960-894X, 5 p.Article

Inverse Agonist of Nuclear Receptor ERRγ Mediates Antidiabetic Effect Through Inhibition of Hepatic GluconeogenesisKIM, Don-Kyu; GANG, Gil-Tae; CHEOL SOO CHOI et al.Diabetes (New York, NY). 2013, Vol 62, Num 9, pp 3093-3102, issn 0012-1797, 10 p.Article

Ac His1 [D-Phe2, K15, R16, L27] VIP (3-7)/GRF (8-27) - a VPAC1 receptor antagonist: is an inverse agonist on two constitutively active truncated VPAC1 receptorsVERTONGEN, Pascale; LANGLET, Christelle; LANGER, Ingrid et al.Peptides (New York, NY. 1980). 2004, Vol 25, Num 11, pp 1943-1949, issn 0196-9781, 7 p.Article

Future trends : A new generation of retinoids. DiscussionCHANDRARATNA, R. A. S.Journal of the American Academy of Dermatology. 1998, Vol 39, Num 4, pp S149-S152, issn 0190-9622, 2Conference Paper

Negative antagonists promote as inactive conformation of the β2-adrenergic receptorSAMAMA, P; GANG PEI; COSTA, T et al.Molecular pharmacology. 1994, Vol 45, Num 3, pp 390-394, issn 0026-895XArticle

Investigation of the mechanism of agonist and inverse agonist action at D2 dopamine receptorsROBERTS, David J; HONG LIN; STRANGE, Philip G et al.Biochemical pharmacology. 2004, Vol 67, Num 9, pp 1657-1665, issn 0006-2952, 9 p.Article

Substituted phenoxypropyl-(R)-2-methylpyrrolidine aminomethyl ketones as histamine-3 receptor inverse agonistsZULLI, Allison L; AIMONE, Lisa D; MATHIASEN, Joanne R et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 8, pp 2807-2810, issn 0960-894X, 4 p.Article

Antibodies as pharmacologic tools for studies on the regulation of energy balanceHOFBAUER, Karl G; LECOURT, Anne-Catherine; PETER, Jean-Christophe et al.Nutrition (Burbank, Los Angeles County, Calif.). 2008, Vol 24, Num 9, pp 791-797, issn 0899-9007, 7 p.Conference Paper

Heterologous desensitization is evoked by both agonist and antagonist stimulation of the human 5-HT7 serotonin receptorKROBERT, Kurt A; ANDRESSEN, Kjetil Wessel; LEVY, Finn Olav et al.European journal of pharmacology. 2006, Vol 532, Num 1-2, pp 1-10, issn 0014-2999, 10 p.Article

Na+ modulation, inverse agonism, and anorectic potency of 4-phenylpiperidine opioid antagonistsEMMERSON, Paul J; MCKINZIE, Jamie H; SURFACE, Peggy L et al.European journal of pharmacology. 2004, Vol 494, Num 2-3, pp 121-130, issn 0014-2999, 10 p.Article

Effects of the benzodiazepine inverse agonist RO19-4603 alone and in combination with the benzodiazepine receptor antagonists flumazenil, ZK 93426 and CGS 8216, on ethanol intake in alcohol-preferring (P) ratsJUNE, H. L; GREENE, T. L; LUMENG, L et al.Brain research. 1996, Vol 734, Num 1-2, pp 19-34, issn 0006-8993Article

Neurosteroid pregnenolone induces sleep-EEG changes in man compatible with inverse agonistic GABAA-receptor modulationSTEIGER, A; TRACHSEL, L; GULDNER, J et al.Brain research. 1993, Vol 615, Num 2, pp 267-274, issn 0006-8993Article

Stimulant effect of the β-carboline FG 7142 in the open-field testBRUHWYLER, J; CHLEIDE, E; HOUBEAU, G et al.European journal of pharmacology. 1991, Vol 200, Num 1, pp 183-185, issn 0014-2999, 3 p.Article

Functional in vivo correlates of the benzodiazepine agonist-inverse agonist continuumGARDNER, C. R.Progress in neurobiology. 1988, Vol 31, Num 6, pp 425-476, issn 0301-0082Article

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