au.\*:("JACOBSON, A. E")
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The LMC delta opioid recognition pharmacophore : Comparison of SNC80 and oxymorphindoleCOOP, A; JACOBSON, A. E.Bioorganic & medicinal chemistry letters (Print). 1999, Vol 9, Num 3, pp 357-362, issn 0960-894XArticle
Probes for narcotic receptor mediated phenomena. 26. Synthesis and biological evaluation of diarylmethylpiperazines and diarylmethylpiperidines as novel, nonpeptidic δ opioid receptor ligandsXIAOYAN ZHANG; RICE, K. C; PORRECA, F et al.Journal of medicinal chemistry (Print). 1999, Vol 42, Num 26, pp 5455-5463, issn 0022-2623Article
Phencyclidine binds to blood platelets with high affinity and specially inhibits their activation by adrenalineJAMIESON, G. A; AGRAWAL, A. K; GRECO, N. J et al.Biochemical journal (London. 1984). 1992, Vol 285, pp 35-39, issn 0264-6021, 1Article
Enantioselective kappa opioid binding sites on the macrophage cell line, P388d1CARR, D. J; DECOSTA, B. R; JACOBSON, A. E et al.Life sciences (1973). 1991, Vol 49, Num 1, pp 45-51, issn 0024-3205Article
Preliminary ligand binding data for subtypes of the dalta opioid receptor in rat brain membranesHENG XU; QING NI; JACOBSON, A. E et al.Life sciences (1973). 1991, Vol 49, Num 18, pp PL.141-PL146, issn 0024-3205Article
The potent opioid agonist, (+)-cis-3-methylfentanyl binds pseudoirreversibly to the opioid receptor complex in vitro and in vivo : evidence for a novel mechanism of actionBAND, L; HENG XU; BYKOV, V et al.Life sciences (1973). 1990, Vol 47, Num 24, pp 2231-2240, issn 0024-3205, 10 p.Article
Very long-acting narcotic antagonists: the 14β-p-substituted cinnamoylaminomorphinones and their partial mu agonist codeinone relativesACETO, M. D; BOWMAN, E. R; MAY, E. L et al.Arzneimittel-Forschung. 1989, Vol 39, Num 5, pp 570-575, issn 0004-4172Article
Pharmacological activities of optically pure enantiomers of the κ opioid agonist, U50,488, and its cis diastereomer: evidence for three κ receptor subtypesROTHMAN, R. B; FRANCE, C. P; BYKOV, V et al.European journal of pharmacology. 1989, Vol 167, Num 3, pp 345-353, issn 0014-2999Article
Tritiated-6-beta-fluoro-6-desoxy-oxymorphone ([3H] FOXY): a new ligand and photoaffinity probe for the MU opioid receptorsROTHMAN, R. B; BYKOV, V; RICE, K. C et al.Neuropeptides (Edinburgh). 1988, Vol 11, Num 1, pp 1-6, issn 0143-4179Article
Intracerebroventricular administration of superfit and its enantiomer to rats: evidence for in vivo acylation of [3H] DADL binding sitesROTHMAN, R. B; LONG, J. B; BYKOV, V et al.Neuropeptides (Edinburgh). 1987, Vol 9, Num 3, pp 207-210, issn 0143-4179Article
Enantiomeric and diastereomeric dioxadrols: behavioral, biochemical and chemical determination of the configuration necessary for phencyclidine-like propertiesJACOBSON, A. E; HARRISON, E. A. JR; MATTSON, M. V et al.The Journal of pharmacology and experimental therapeutics. 1987, Vol 243, Num 1, pp 110-117, issn 0022-3565Article
Metaphit, a proposed phencyclidine (PCP) antagonist, prevents PCP-induced locomotor behavior through mechanisms unrelated to specific blockade of PCP receptorsFRENCH, E. D; JACOBSON, A. E; RICE, K. C et al.European journal of pharmacology. 1987, Vol 140, Num 3, pp 267-274, issn 0014-2999Article
Phencyclidine (PCP)-like discriminative stimulus effects of metaphit and of 2-amino-5-phosphonovalerate in pigeons: generality across different training doses of PCPKOEK, W; WOODS, J. H; JACOBSON, A. E et al.Psychopharmacologia. 1987, Vol 93, Num 4, pp 437-442, issn 0033-3158Article
Morphine tolerance increases μ-noncompatitive δ binding sitesROTHMAN, R. B; DANKS, J. A; JACOBSON, A. E et al.European journal of pharmacology. 1986, Vol 124, Num 1-2, pp 113-119, issn 0014-2999Article
Probes for narcotic receptor mediated phenomena. XII: cis-(+)-3-Methylfentanyl isothiocyanate, a potent site-directed acylating agent for δ opioid receptors. Synthesis, absolute configuration, and receptor enantioselectivityBURKE, T. R. JR; JACOBSON, A. E; RICE, K. C et al.Journal of medicinal chemistry (Print). 1986, Vol 29, Num 6, pp 1087-1093, issn 0022-2623Article
A specific alkylating ligand for phenyclidine (PCP) receptors antagonizes PCP behavioral effectsCONTRERAS, P. C; RAFFERTY, M. F; LESSOR, R. A et al.European journal of pharmacology. 1985, Vol 111, Num 3, pp 405-406, issn 0014-2999Article
Pharmacological actions of the racemic and the enantiomeric 1,4-dimethyl-10-hydroxy-2,3,4,5,6,7-hexahydro-1,6-methano-1H-4-benzazonines (C-homobenzomorphans)ACETO, M. D; HARRIS, L. S; WOODS, J. H et al.Japanese journal of pharmacology. 1985, Vol 39, Num 1, pp 7-19, issn 0021-5198Article
Discriminative stimulus effects of reversible and irreversible opiate agonists: morphine, oxymorphazone and buprenorphineFRANCE, C. P; JACOBSON, A. E; WOODS, J. H et al.The Journal of pharmacology and experimental therapeutics. 1984, Vol 230, Num 3, pp 652-657, issn 0022-3565Article
Stereospecificity of 4,5-epoxymorphinan binding to the λ site in rat brainYU, V. C; JACOBSON, A. E; RICE, K. C et al.European journal of pharmacology. 1984, Vol 101, Num 1-2, pp 161-162, issn 0014-2999Article
9α- and 9β-HydroxyphenylmorphansAWAYA, H; MAY, E. L; JACOBSON, A. E et al.Journal of pharmaceutical sciences. 1984, Vol 73, Num 12, pp 1867-1868, issn 0022-3549Article
Agonist-antagonist actions and stereoselectivity of optical pairs of some N-substituted α-N-normetazocinesACETO, M. D; MAY, E. L; HARRIS, L. S et al.Journal of pharmaceutical sciences. 1984, Vol 73, Num 12, pp 1864-1866, issn 0022-3549Article
Antipodal α-N-(methyl through decyl)-N-normetazocines (5,9α-dimethyl-2'-hydroxy-6,7-benzomorphans) : in vitro and in vivo propertiesMAY, E. L; ACETO, M. D; BOWMAN, E. R et al.Journal of medicinal chemistry (Print). 1994, Vol 37, Num 20, pp 3408-3418, issn 0022-2623Article
Metaphit-induced audiogenic seizures in mice. I: Pharmacologic characterizationDEBLER, E. A; LIPOVAC, M. N; LAJTHA, A et al.Epilepsia (Copenhagen). 1993, Vol 34, Num 2, pp 201-210, issn 0013-9580Article
Synthesis and binding properties of MK-801 isothiocyanates ; (+)-3-isothiocyanato-5-methyl-10,11-dihydro-5-dibenzo[a,d]cyclohepten-5,10-imine hydrochloride : a new, potent and selective electrophilic affinity ligand for the NMDA receptor-coupled phencyclidine binding siteLINDERS, J. T. M; MONN, J. A; MATTSON, M. V et al.Journal of medicinal chemistry (Print). 1993, Vol 36, Num 17, pp 2499-2507, issn 0022-2623Article
Interaction of endogenous opioid peptides and other drugs with four kappa opioid binding sites in guinea pig brainROTHMAN, R. B; BYKOV, V; DE COSTA, B. R et al.Peptides (New York, NY. 1980). 1990, Vol 11, Num 2, pp 311-331, issn 0196-9781Article