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Analytical challenges in drug counterfeiting and falsification—The NMR approachHOLZGRABE, Ulrike; MALET-MARTINO, Myriam.Journal of pharmaceutical and biomedical analysis. 2011, Vol 55, Num 4, pp 679-687, issn 0731-7085, 9 p.Article

Fluorouracil prodrugs for the treatment of proliferative vitreoretinopathy: formulation in silicone oil and in vitro release of fluorouracilJOLIMAITRE, Pascale; MALET-MARTINO, Myriam; MARTINO, Robert et al.International journal of pharmaceutics. 2003, Vol 259, Num 1-2, pp 181-192, issn 0378-5173, 12 p.Article

ETUDE DE MEDICAMENTS ANTICANCEREUX PAR RESONANCE MAGNETIQUE NUCLEAIRE 31P, 19F, 13C et 1H : STABILITE ET METABOLISME DE L'ISOPHOSPHORAMIDE MOUTARDE ET DU GLUFOSFAMIDE, AGENTS PHOSPHORES ; TOXICITE ET METABOLISME DU 5-FLUOROURACILE ET DE LA CAPECITABINE, MEDICAMENTS FLUORES = STUDY OF ANTICANCER DRUGS BY 31P, 19F, 13C AND 1H NUCLEAR MAGNETIC RESONANCE : - STABILITY AND METABOLISM OF ISOPHOSPHORAMIDE MUSTARD AND GLUFOSFAMIDE, PHOSPHORYLATED AGENTS ; - TOXICITY AND METABOLISM OF 5-FLUOROURACIL AND CAPECITABINE, FLUORINATED DRUGSBreil, Stephane; Malet Martino, Myriam.1999, 165 p.Thesis

Métabolisme hépatique du 5-fluorouracile par résonance magnétique nucléaire du fluor-19 = 5-fluorouracil hepatic metabolism by fluorine-19 nuclear magnetic resonanceLongo Cabanac, Sophie; Malet-Martino, Myriam.1991, 294 p.Thesis

Isolation of an unknown metabolite of capecitabine, an oral 5-fluorouracil prodrug, and its identification by nuclear magnetic resonance and liquid chromatography-tandem mass spectrometry as a glucuroconjugate of 5'-deoxy-5-fluorocytidine, namely 2'-(β-D-glucuronic acid)-5'-deoxy-5-fluorocytidineDESMOULIN, Franck; GILARD, Véronique; MARTINO, Robert et al.Journal of chromatography. B. 2003, Vol 792, Num 2, pp 323-332, issn 1570-0232, 10 p.Article

Generic ciprofloxacin tablets contain the stated amount of drug and different impurity profiles : A 19F, 1H and DOSY NMR analysisTREFI, Saleh; GILARD, Véronique; MALET-MARTINO, Myriam et al.Journal of pharmaceutical and biomedical analysis. 2007, Vol 44, Num 3, pp 743-754, issn 0731-7085, 12 p.Article

Metabolism of capecitabine, an oral fluorouracil prodrug: 19F NMR studies in animal models and human urineDESMOULIN, Franck; GILARD, Véronique; MALET-MARTINO, Myriam et al.Drug metabolism and disposition. 2002, Vol 30, Num 11, pp 1221-1229, issn 0090-9556, 9 p.Article

Interest of fluorine-19 nuclear magnetic resonance spectroscopy in the detection, identification and quantification of metabolites of anticancer and antifungal fluoropyrimidine drugs in human biofluidsMARTINO, Robert; GILARD, Véronique; DESMOULIN, Franck et al.Chemotherapy (Basel). 2006, Vol 52, Num 5, pp 215-219, issn 0009-3157, 5 p.Conference Paper

Quality assessment of fluoxetine and fluvoxamine pharmaceutical formulations purchased in different countries or via the Internet by 19F and 2D DOSY 1H NMRTREFI, Saleh; GILARD, Véronique; BALAYSSAC, Stéphane et al.Journal of pharmaceutical and biomedical analysis. 2008, Vol 46, Num 4, pp 707-722, issn 0731-7085, 16 p.Article

Fluorine-19 or phosphorus-31 NMR spectroscopy : A suitable analytical technique for quantitative in vitro metabolic studies of fluorinated or phosphorylated drugsMARTINO, Robert; GILARD, Véronique; DESMOULIN, Franck et al.Journal of pharmaceutical and biomedical analysis. 2005, Vol 38, Num 5, pp 871-891, issn 0731-7085, 21 p.Article

Identification of a novel sildenafil analogue in an adulterated herbal supplementVAYSSE, Julie; GILARD, Veronique; BALAYSSAC, Stéphane et al.Journal of pharmaceutical and biomedical analysis. 2012, Vol 59, pp 58-66, issn 0731-7085, 9 p.Article

Identification of new aqueous chemical degradation products of isophosphoramide mustardBREIL, Stéphane; MARTINO, Robert; GILARD, Véronique et al.Journal of pharmaceutical and biomedical analysis. 2001, Vol 25, Num 3-4, pp 669-678, issn 0731-7085Article

Analysis of herbal dietary supplements for sexual performance enhancement: First characterization of propoxyphenyl-thiohydroxyhomosildenafil and identification of sildenafil, thiosildenafil, phentolamine and tetrahydropalmatine as adulterantsBALAYSSAC, Stephane; GILARD, Veronique; ZEDDE, Chantal et al.Journal of pharmaceutical and biomedical analysis. 2012, Vol 63, pp 135-150, issn 0731-7085, 16 p.Article

Analysis of illegally manufactured formulations of tadalafil (Cialis®) by 1H NMR, 2D DOSY 1H NMR and Raman spectroscopyTREFI, Saleh; ROUTABOUL, Corinne; HAMIEH, Saleh et al.Journal of pharmaceutical and biomedical analysis. 2008, Vol 47, Num 1, pp 103-113, issn 0731-7085, 11 p.Article

2D and 3D DOSY 1H NMR, a useful tool for analysis of complex mixtures: Application to herbal drugs or dietary supplements for erectile dysfunctionBALAYSSAC, Stéphane; TREFI, Saleh; GILARD, Véronique et al.Journal of pharmaceutical and biomedical analysis. 2009, Vol 50, Num 4, pp 602-612, issn 0731-7085, 11 p.Conference Paper

Stability of commercial solutions of 5-fluorouracil for continuous infusion in an ambulatory pumpFOURNET, Alexandra; GILARD, Véronique; MALET-MARTINO, Myriam et al.Cancer chemotherapy and pharmacology. 2000, Vol 46, Num 6, pp 501-506, issn 0344-5704Article

Synthesis of lipophilic dimeric C-7/C-7-linked ciprofloxacin and C-6/C-6-linked levofloxacin derivatives. Versatile in vitro biological evaluations of monomeric and dimeric fluoroquinolone derivatives as potential antitumor, antibacterial or antimycobacterial agentsAZEMA, Joëlle; GUIDETTI, Brigitte; KOROLYOV, Alexander et al.European journal of medicinal chemistry. 2011, Vol 46, Num 12, pp 6025-6038, issn 0223-5234, 14 p.Article

Usefulness of in vitro 1H magnetic resonance spectroscopy for the characterization of primary brain tumors : Report of two casesSABATIER, Jean; ROBERT, Olivier; DELISLE, Marie-Bernadette et al.Stereotactic and functional neurosurgery. 2005, Vol 83, Num 2-3, pp 122-127, issn 1011-6125, 6 p.Article

Interaction mechanism between caffeine and polyphenols in infusions of Camellia sinensis leavesCOUZINET-MOSSION, Aurélie; BALAYSSAC, Stéphane; GILARD, Véronique et al.Food chemistry. 2010, Vol 119, Num 1, pp 173-181, issn 0308-8146, 9 p.Article

Étude critique de l'utilisation de la RMN HR-MAS pour l'analyse des tissus biologiques = HR-MAS NMR analysis of biological tissues : a critical reportDESMOULIN, Franck; BON, Delphine; MARTINO, Robert et al.Comptes rendus. Chimie. 2008, Vol 11, Num 4-5, pp 423-433, issn 1631-0748, 11 p.Conference Paper

Combining Two-Dimensional Diffusion-Ordered Nuclear Magnetic Resonance Spectroscopy, Imaging Desorption Electrospray Ionization Mass Spectrometry, and Direct Analysis in Real-Time Mass Spectrometry for the Integral Investigation of Counterfeit PharmaceuticalsNYADONG, Leonard; HARRIS, Glenn A; BALAYSSAC, Stéphane et al.Analytical chemistry (Washington). 2009, Vol 81, Num 12, pp 4803-4812, issn 0003-2700, 10 p.Article

Inactivation of the HIF-1α/PDK3 Signaling Axis Drives Melanoma toward Mitochondrial Oxidative Metabolism and Potentiates the Therapeutic Activity of Pro-OxidantsKLUZA, Jérome; CORAZAO-ROZAS, Paola; CORROYER-DULMONT, Aurélien et al.Cancer research (Chicago, Ill.). 2012, Vol 72, Num 19, pp 5035-5047, issn 0008-5472, 13 p.Article

Novel lipophilic 7H-pyrido[1,2,3-de]-1,4-benzoxazine-6-carboxylic acid derivatives as potential antitumor agents: Improved synthesis and in vitro evaluationKOROLYOV, Alexander; DORBES, Sandra; MALET-MARTINO, Myriam et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 24, pp 8537-8548, issn 0968-0896, 12 p.Article

7-((4-Substituted)piperazin-1-yl) derivatives of ciprofloxacin: Synthesis and in vitro biological evaluation as potential antitumor agentsAZEMA, Joëlle; GUIDETTI, Brigitte; DEWELLE, Janique et al.Bioorganic & medicinal chemistry. 2009, Vol 17, Num 15, pp 5396-5407, issn 0968-0896, 12 p.Article

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