Design, synthesis, structural studies, biological evaluation, and computational simulations of novel potent AT₁ angiotensin II receptor antagonists based on the 4-phenylquinoline structureCAPPELLI, Andrea; MOHR, Gal La; DE BENEDETTI, Pier G et al.Journal of medicinal chemistry (Print). 2004, Vol 47, Num 10, pp 2574-2586, issn 0022-2623, 13 p.Article

Further studies on imidazo[4,5-b]pyridine AT₁ angiotensin II receptor antagonists. Effects of the transformation of the 4-phenylquinoline backbone into 4-phenylisoquinolinone or 1-phenylindene scaffoldsCAPPELLI, Andrea; PERICOT MOHR, Galla; VALOTI, Massimo et al.Journal of medicinal chemistry (Print). 2006, Vol 49, Num 22, pp 6451-6464, issn 0022-2623, 14 p.Article

Structure-affinity relationship studies on arylpiperazine derivatives related to quipazine as serotonin transporter ligands. Molecular basis of the selectivity SERT/5HT₃ receptorCAPPELLI, Andrea; GIULIANI, Germano; GALLELLI, Andrea et al.Bioorganic & medicinal chemistry. 2005, Vol 13, Num 10, pp 3455-3460, issn 0968-0896, 6 p.Article

Anthranilic acid based CCK₁ receptor antagonists : preliminary investigation on their second touch pointVARNAVAS, Antonio; LASSIANI, Lucia; VALENTA, Valentina et al.European journal of medicinal chemistry. 2005, Vol 40, Num 6, pp 563-581, issn 0223-5234, 19 p.Article

Anthranilic acid based CCK₁ antagonists: the 2-indole moiety may represent a needle according to the recent homonymous conceptVARNAVAS, Antonio; LASSIANI, Lucia; VALENTA, Valentina et al.European journal of medicinal chemistry. 2004, Vol 39, Num 1, pp 85-97, issn 0223-5234, 13 p.Article

Anthranilic acid derivatives : A new class of non-peptide CCK₁ receptor antagonistsVARNAVAS, Antonio; LASSIANI, Lucia; VALENTA, Valentina et al.Bioorganic & medicinal chemistry. 2003, Vol 11, Num 5, pp 741-751, issn 0968-0896, 11 p.Article

Novel potent 5-HT₃ receptor ligands based on the pyrrolidone structure. effects of the quaternization of the basic nitrogen on the interaction with 5-HT₃ receptorCAPPELLI, Andrea; GALLELLI, Andrea; GIORGI, Gianluca et al.Bioorganic & medicinal chemistry. 2002, Vol 10, Num 8, pp 2681-2691, issn 0968-0896Article

Multivalent Supramolecular Dendrimer-Based DrugsGALEAZZI, Simone; HERMANS, Thomas M; CAPPELLI, Andrea et al.Biomacromolecules. 2010, Vol 11, Num 1, pp 182-186, issn 1525-7797, 5 p.Article

Anthranilic acid based CCK₁ receptor antagonists : Blocking the receptor with the same 'mords' of the endogenous ligandLASSIANI, Lucia; PAVAN, Michela V; BERTI, Federico et al.Bioorganic & medicinal chemistry. 2009, Vol 17, Num 6, pp 2336-2350, issn 0968-0896, 15 p.Article

Design, Synthesis, and Biological Evaluation of AT₁ Angiotensin II Receptor Antagonists Based on the Pyrazolo[3,4-b]pyridine and Related Heteroaromatic Bicyclic SystemsCAPPELLI, Andrea; NANNICINI, Chiara; GIORDANI, Antonio et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 7, pp 2137-2146, issn 0022-2623, 10 p.Article

Further studies on the interaction of the 5-hydroxytryptamine₃ (5-HT₃) receptor with arylpiperazine ligands. Development of a new 50-HT₃ receptor ligand showing potent acetylcholinesterase inhibitory propertiesCAPPELLI, Andrea; GALLELLI, Andrea; MANINI, Monica et al.Journal of medicinal chemistry (Print). 2005, Vol 48, Num 10, pp 3564-3575, issn 0022-2623, 12 p.Article

Novel potent 5-HT₃ receptor ligands based on the pyrrolidone structure: Synthesis, biological evaluation, and computational rationalization of the ligand-receptor interaction modalitiesCAPPELLI, Andrea; ANZINI, Maurizio; GHELARDINI, Carla et al.Bioorganic & medicinal chemistry. 2002, Vol 10, Num 3, pp 779-801, issn 0968-0896Article