Inhibition by 5-HT of forskolin-induced cAMP formation in the renal opossum epithelial cell line OK : mediation by a 5-HT_1B like receptor and antagonism by methiothepinPAUWELS, P. J; PALMIER, C.Neuropharmacology. 1994, Vol 33, Num 1, pp 67-75, issn 0028-3908Article

Functional effects of the 5-HT_1D receptor antagonist GR 127,935 at human 5-HT_1Dα, 5-HT_1Dβ, 5-HT_1A and opossum 5-HT_1B receptorsPAUWELS, P. J; PALMIER, C.European journal of pharmacology. Molecular pharmacology section. 1995, Vol 290, Num 2, pp 95-103, issn 0922-4106Article

Role of fructose 2,6-bisphosphate in the regulation of glycolysis in various types of cultivated brain cellPAUWELS, P. J; TROUET, A.Neuroscience letters. 1984, Vol 46, Num 2, pp 173-177, issn 0304-3940Article

Recombinant saphenous vein 5-HT_1B receptors of the rabbit : comparative pharmacology with human 5-HT_1B receptorsWURCH, T; PALMIER, C; COLPAERT, F. C et al.British journal of pharmacology. 1997, Vol 120, Num 1, pp 153-159, issn 0007-1188Article

Selective antagonism of human 5-HT_1D and 5-HT_1B receptor-mediated responses in stably transfected C6-glial cells by ketanserin and GR 127,935PAUWELS, P. J; COLPAERT, F. C.European journal of pharmacology. 1996, Vol 300, Num 1-2, pp 141-146, issn 0014-2999, 5 p.Article

Comparison of in vitro binding properties of a series of dopamine antagonists and agonists for cloned human dopamine D_2S and D_2L receptors and for D₂ receptors in rat striatal and mesolimbic tissues, using [¹²⁵I] 2'-iodospiperoneLEYSEN, J. E; GOMMEREN, W; MERTENS, J et al.Psychopharmacologia. 1993, Vol 110, Num 1-2, pp 27-36, issn 0033-3158Article

Identifications of 5-hydroxytryptamine_1D binding sites in sheep caudate nucleus membranesPAUWELS, P. J; PALMIER, C; BRILEY, M et al.Biochemical pharmacology. 1993, Vol 46, Num 3, pp 535-538, issn 0006-2952Article

Blockade of nitric oxide formation does not prevent glutamate-induced neurotoxicity in neuronal cultures from rat hippocampusPAUWELS, P. J; LEYSEN, J. E.Neuroscience letters. 1992, Vol 143, Num 1-2, pp 27-30, issn 0304-3940Article

Autoradiography of serotonin 5-HT_1A receptor-activated G proteins in guinea pig brain sections by agonist-stimulated [³⁵S]GTPγS bindingDUPUIS, D. S; PALMIER, C; COLPAERT, F. C et al.Journal of neurochemistry. 1998, Vol 70, Num 3, pp 1258-1268, issn 0022-3042Article

Differentiation between partial agonists and neutral 5-HT_1B antagonists by chemical modulation of 3-[3-(N,N-dimethylamino)propyl]-4-hydroxy-N-[4-(pyridin-4-yl)phenyl]benzamide (GR-55562)LAMOTHE, M; PAUWELS, P. J; BELLIARD, K et al.Journal of medicinal chemistry (Print). 1997, Vol 40, Num 22, pp 3542-3550, issn 0022-2623Article

How efficacious are 5-HT_1B/D receptor ligands : An answer from GTPγS binding studies with stably transfected C6-glial cell linesPAUWELS, P. J; TARDIF, S; PALMIER, C et al.Neuropharmacology. 1997, Vol 36, Num 4-5, pp 499-512, issn 0028-3908Article

Synthesis and serotonergic activity of arylpiperazide derivatives of serotonin : potent agonists for 5-HT_1D receptorsPEREZ, M; FOURRIER, C; SIGOGNEAU, I et al.Journal of medicinal chemistry (Print). 1995, Vol 38, Num 18, pp 3602-3607, issn 0022-2623Article

Expression of human metallothionein-III confers protection against serum-free exposure of stably transfected Chinese hamster ovary CHO-K1 cellsAMOUREUX, M.-C; WURCH, T; PAUWELS, P. J et al.Neuroscience letters. 1995, Vol 201, Num 1, pp 61-64, issn 0304-3940Article

Activity of serotonin (5-HT) receptor agonists, partial agonists and antagonists at cloned human 5-HT_1A receptors that are negatively coupled to adenylate cyclase in permanently transfected HeLa cellsPAUWELS, P. J; VAN GOMPEL, P; LEYSEN, J. E et al.Biochemical pharmacology. 1993, Vol 45, Num 2, pp 375-383, issn 0006-2952Article

Disparate ligand-mediated Ca²⁺ responses by wild-type, mutant Ser²⁰⁰ Ala and Ser²⁰⁴ Ala α_2A-adrenoceptor : G_α15 fusion proteins : evidence for multiple ligand-activation binding sitesPAUWELS, P. J; COLPAERT, F. C.British journal of pharmacology. 2000, Vol 130, Num 7, pp 1505-1512, issn 0007-1188Article

G-protein activation by putative antagonists at mutant Thr³⁷³Lys α_2A adrenergic receptorsWURCH, T; COLPAERT, F. C; PAUWELS, P. J et al.British journal of pharmacology. 1999, Vol 126, Num 4, pp 939-948, issn 0007-1188Article

Present and future of 5-HT receptor agonists as antimigraine drugsPAUWELS, P. J; JOHN, G. W.Clinical neuropharmacology. 1999, Vol 22, Num 3, pp 123-136, issn 0362-5664Article

The 5-HT_1D receptor antagonist GR 127,935 is an agonist at cloned human 5-HT_1Dα receptor sitesPAUWELS, P. J; COLPAERT, F. C.Neuropharmacology. 1995, Vol 34, Num 2, pp 235-237, issn 0028-3908Article

Heterogeneous ligand-mediated Ca⁺⁺ responses at wt and mutant α_2A-adrenoceptors suggest multiple ligand activation binding sites at the α_2A-adrenoceptorPAUWELS, P. J; COLPAERT, F. C.Neuropharmacology. 2000, Vol 39, Num 11, pp 2101-2111, issn 0028-3908Article

Cultivation of rat cerebellar cells under conditions of optimal oxygen supplyPAUWELS, P. J; ABARCA, J; TROUET, A et al.Neuroscience letters. 1983, Vol 43, Num 2-3, pp 309-314, issn 0304-3940Article

Large-amplitude 5-HT_1A receptor activation: a new mechanism of profound, central analgesiaCOLPAERT, F. C; TARAYRE, J. P; VACHER, B et al.Neuropharmacology. 2002, Vol 43, Num 6, pp 945-958, issn 0028-3908, 14 p.Article

Magnitude of 5-HT_1B and 5-HT_1A receptor activation in guinea-pig and rat brain : Evidence from sumatriptan dimer-mediated [³⁵S]GTPγS binding responsesDUPUIS, D. S; PEREZ, M; HALAZY, S et al.Molecular brain research. 1999, Vol 67, Num 1, pp 107-123, issn 0169-328XArticle

Pharmacological analysis of G-protein activation mediated by guinea-pig recombinant 5-HT_1B receptors in C6-glial cells : similarities with the human 5-HT_1B receptorPAUWELS, P. J; WURCH, T; PALMIER, C et al.British journal of pharmacology. 1998, Vol 123, Num 1, pp 51-62, issn 0007-1188Article

Design and synthesis of new potent, silent 5-HT_1A antagonists by covalent coupling of aminopropanol derivatives with selective serotonin reuptake inhibitorsPEREZ, M; PAUWELS, P. J; PALLARD-SIGOGNEAU, I et al.Bioorganic & medicinal chemistry letters (Print). 1998, Vol 8, Num 23, pp 3423-3428, issn 0960-894XArticle

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