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au.\*:("PAVLYUKOVETS, Vladimir A")

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Conformationally constrained analogues of diacylglycerol (DAG). 27. modulation of membrane translocation of protein kinase C (PKC) isozymes α and δ by diacylglycerol lactones (DAG-lactones) containing rigid-rod acyl groupsMALOLANARASIMHAN, Krishnan; KEDEI, Noemi; BLUMBERG, Peter M et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 5, pp 962-978, issn 0022-2623, 17 p.Article

Non-vanillyl resiniferatoxin analogues as potent and metabolically stable transient receptor potential vanilloid 1 agonistsCHOI, Hyun-Kyung; CHOI, Sun; TRAN, Richard et al.Bioorganic & medicinal chemistry. 2009, Vol 17, Num 2, pp 690-698, issn 0968-0896, 9 p.Article

Stereospecific High-affinity TRPV1 Antagonists : Chiral N-(2-Benzyl-3-pivaloyloxypropyl) 2-[4-(methylsulfonylamino)phenyl]propionamide AnaloguesRYU, Hyungchul; JIN, Mi-Kyoung; TRAN, Richard et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 1, pp 57-67, issn 0022-2623, 11 p.Article

Structure―activity relationships and molecular modeling of the N-(3-pivaloyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl] thiourea template for TRPV1 antagonismBHONDWE, Rahul S; DONG WOOK KANG; BLUMBERG, Peter M et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 11, pp 3656-3660, issn 0960-894X, 5 p.Article

Analysis of structure-activity relationships for the 'B-region' of N-(4-t-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl ]- thiourea analogues as TRPV1 antagonistsLEE, Jeewoo; JIN, Mi-Kyoung; KIM, Sung-Eun et al.Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 18, pp 4143-4150, issn 0960-894X, 8 p.Article

2-(4-Methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure―activity relationships in the B and C-regionsWEI SUN; KELIANG LIU; PEARCE, Larry V et al.Bioorganic & medicinal chemistry. 2012, Vol 20, Num 3, pp 1310-1318, issn 0968-0896, 9 p.Article

The SAR analysis of TRPV1 agonists with the α-methylated B-regionCHO, Yongsung; MYEONG SEOP KIM; HO SHIN KIM et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 16, pp 5227-5231, issn 0960-894X, 5 p.Article

Halogenation of 4-hydroxy/amino-3-methoxyphenyl acetamide TRPV1 agonists showed enhanced antagonism to capsaicinDONG WOOK KANG; YONG SOO KIM; KWANG SU LIM et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 22, pp 8092-8105, issn 0968-0896, 14 p.Article

α-Substituted N-(4 -tert-butylbenzyl ) -N'-[4 -(methylsulfonylamino )-benzyl]thiourea analogues as potent and stereospecific TRPV1 antagonistsCHUNG, Jae-Uk; SU YEON KIM; CHOI, Sun et al.Bioorganic & medicinal chemistry. 2007, Vol 15, Num 18, pp 6043-6053, issn 0968-0896, 11 p.Article

Analysis of structure-activity relationships for the 'A-region' of N-(4-t-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues as TRPV1 antagonistsLEE, Jeewoo; KANG, Sang-Uk; MIN, Kyung-Hoon et al.Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 18, pp 4136-4142, issn 0960-894X, 7 p.Article

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