Synthesis and characterization of [³H]-SN56, a novel radioligand for the σ₁ receptorFISHBACK, James A; MESANGEAU, Christophe; POUPAERT, Jacques H et al.European journal of pharmacology. 2011, Vol 653, Num 1-3, pp 1-7, issn 0014-2999, 7 p.Article

Interactions between 3,4-methylenedioxymethamphetamine and σ₁ receptorsBRAMMER, Matthew K; GILMORE, Deborah L; MATSUMOTO, Rae R et al.European journal of pharmacology. 2006, Vol 553, Num 1-3, pp 141-145, issn 0014-2999, 5 p.Article

CB-64D and CB-184 : ligands with high ₂ receptor affinity and subtype selectivityBOWEN, W. D; BERTHA, C. M; VILNER, B. J et al.European journal of pharmacology. 1995, Vol 278, Num 3, pp 257-260, issn 0014-2999Article

High affinity of sigma₁-binding sites for sterol isomerization inhibitors : evidence for a pharmacological relationship with the yeast sterol C₈-C₇ isomeraseMOEBIUS, F. F; REITER, R. J; HANNER, M et al.British journal of pharmacology. 1997, Vol 121, Num 1, pp 1-6, issn 0007-1188Article

The dopamine stabilizers ACR16 and (―)-OSU6162 display nanomolar affinities at the σ-1 receptorSAHLHOLM, K; ARHEM, P; FUXE, K et al.Molecular psychiatry. 2013, Vol 18, Num 1, pp 12-14, issn 1359-4184, 3 p.Article

Thioxanthene-derived analogs as σ₁ receptor ligandsGLENNON, Richard A; ISMAIEL, Abd M; ABLORDEPPEY, Seth et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 9, pp 2217-2220, issn 0960-894X, 4 p.Article

Sigma receptors and cancer: Possible involvement of ion channelsAYDAR, Ebru; PALMER, Christopher P; DJAMGOZ, Mustafa B. A et al.Cancer research (Baltimore). 2004, Vol 64, Num 15, pp 5029-5035, issn 0008-5472, 7 p.Article

The Sigma Enigma : Can Sigma Receptors Provide a Novel Target for Disorders of Mood and Cognition?STAHL, Stephen M.The Journal of clinical psychiatry. 2008, Vol 69, Num 11, pp 1673-1674, issn 0160-6689, 2 p.Article

Classes of Sigma₂ (σ₂) Receptor Ligands: Structure Affinity Relationship (SAfiR) Studies and Antiproliferative Activity : Sigma Receptor Research: Progress Towards Diagnostic and Therapeutic Uses of Sigma LigandsABATE, Carmen; PERRONE, Roberto; BERARDI, Francesco et al.Current pharmaceutical design (Print). 2012, Vol 18, Num 7, pp 938-949, issn 1381-6128, 12 p.Article

Exploration of ring size in a series of cyclic vicinal diamines with σ₁ receptor affinityMOUSSA, Iman A; BANISTERA, Samuel D; MANOLI, Miral et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 17, pp 5493-5497, issn 0960-894X, 5 p.Article

(+)-SKF-10,047 and dextromethorphan ameliorate conditioned fear stress through the activation of phenytoin-regulated σ₁ sitesKAMEI, H; KAMEYAMA, T; NABESHIMA, T et al.European journal of pharmacology. 1996, Vol 299, Num 1-3, pp 21-28, issn 0014-2999Article

Binding properties of SA4503, a novel and selective σ₁ receptor agonistMATSUNO, K; NAKAZAWA, M; OKAMOTO, K et al.European journal of pharmacology. 1996, Vol 306, Num 1-3, pp 271-280, issn 0014-2999, 9 p.Article

[³H]1,3-di(2-tolyl) guanidine binds to a σ₂ receptor on Jurkat cell membranes, but σ compounds fail to influence immunomodulatory events in human peripheral blood lymphocytesDEHAVEN-HUDKINS, D. L; DAUBERT, J. D; SAWUTZ, D. G et al.Immunopharmacology (New York). 1996, Vol 35, Num 1, pp 27-39, issn 0162-3109Article

σ₂ Site-mediated inhibition of electrically evoked guinea pig ileum longitudinal muscle/myenteric plexus contractionsKINNEY, G. G; HARRIS, E. W; RAY, R et al.European journal of pharmacology. 1995, Vol 294, Num 2-3, pp 547-553, issn 0014-2999Article

RLH-033, a novel, potent and selective ligand for the σ₁ recognition siteHUDKINS, R. L; MAILMAN, R. B; DEHAVEN-HUDKINS, D. L et al.European journal of pharmacology. 1994, Vol 271, Num 1, pp 235-236, issn 0014-2999Article

7-Azabicyclo[2.2.1]heptane as a scaffold for the development of selective sigma-2 (σ₂) receptor ligandsBANISTER, Samuel D; RENDINA, Louis M; KASSIOU, Michael et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 12, pp 4059-4063, issn 0960-894X, 5 p.Article

Understanding the molecular mechanism of sigma-1 receptors: Towards a hypothesis that sigma-1 receptors are intracellular amplifiers for signal transduction : Rational drug design and the discovery of the 1,2,3-triazolines as a unique class of anticonvulsants and antiischemic agentsSU, Tsung-Ping; HAYASHI, Teruo.Current medicinal chemistry. 2003, Vol 10, Num 20, pp 2073-2080, issn 0929-8673, 8 p.Article

Differences in cytochrome P450 forms involved in the metabolism of N, N-dipropyl-2-[4-methoxy-3-(2-phenylethoxy)phenyl]ethylamine monohydrochloride (NE-100), a novel sigma ligand, in human liver and intestineYAMAMOTO, Takahito; HAGIMA, Naoko; NAKAMURA, Masato et al.Drug metabolism and disposition. 2003, Vol 31, Num 1, pp 60-66, issn 0090-9556, 7 p.Article

Identification of a 27-kDa high affinity phenylalkylamine-binding polypeptide as the σ₁ binding site by photoaffinity labeling and ligand-directed antibodiesMOEBIUS, F. F; BURROWS, G. G; HANNER, M et al.Molecular pharmacology. 1993, Vol 44, Num 5, pp 966-971, issn 0026-895XArticle

Autoradiographic distribution of [³H](+)-pentazocine and [³H]1,3-di-o-tolylguanidine (DTG) binding sites in guinea pig brain : a comparative studyWALKER, J. M; BOWEN, W. D; GOLDSTEIN, S. R et al.Brain research. 1992, Vol 581, Num 1, pp 33-38, issn 0006-8993Article

Synthesis and pharmacological evaluation of potent and enantioselective σ₁ and σ₂ ligandsMARRAZZO, Agostino; PREZZAVENTO, Orazio; PASQUINUCCI, Lorella et al.Il Farmaco (Pavia). 2001, Vol 56, Num 3, pp 181-189, issn 0014-827XConference Paper

(5S)-3-aryl-5-(1-piperidinylmethyl)-2-oxazolidinones, a new class of potential neuroleptics with a high affinity for sigma receptorsPRÜCHER, H; GOTTSCHLICH, R; HAASE, A et al.Bioorganic & medicinal chemistry letters. 1992, Vol 2, Num 2, pp 165-170Article

SN79, a sigma receptor ligand, blocks methamphetamine-induced microglial activation and cytokine upregulationROBSON, Matthew J; TURNER, Ryan C; NASER, Zachary J et al.Experimental neurology (Print). 2013, Vol 247, pp 134-142, issn 0014-4886, 9 p.Article

Molecular mechanisms involving sigma receptor-mediated induction of MCP-1: implication for increased monocyte transmigrationHONGHONG YAO; YANJING YANG; KEE JUN KIM et al.Blood. 2010, Vol 115, Num 23, pp 4951-4962, issn 0006-4971, 12 p.Article

Formalin-induced pain is reduced in σ₁ receptor knockout miceCENDAN, Cruz Miguel; PUJALTE, José Miguel; PORTILLO-SALIDO, Enrique et al.European journal of pharmacology. 2005, Vol 511, Num 1, pp 73-74, issn 0014-2999, 2 p.Article