Synthesis and characterization of [³H]-SN56, a novel radioligand for the σ₁ receptorFISHBACK, James A; MESANGEAU, Christophe; POUPAERT, Jacques H et al.European journal of pharmacology. 2011, Vol 653, Num 1-3, pp 1-7, issn 0014-2999, 7 p.Article

Formalin-induced pain is reduced in σ₁ receptor knockout miceCENDAN, Cruz Miguel; PUJALTE, José Miguel; PORTILLO-SALIDO, Enrique et al.European journal of pharmacology. 2005, Vol 511, Num 1, pp 73-74, issn 0014-2999, 2 p.Article

Involvement of sigma-1 receptor modulation in the antidepressant action of venlafaxineDHIR, Ashish; KULKARNI, S. K.Neuroscience letters. 2007, Vol 420, Num 3, pp 204-208, issn 0304-3940, 5 p.Article

Interactions between 3,4-methylenedioxymethamphetamine and σ₁ receptorsBRAMMER, Matthew K; GILMORE, Deborah L; MATSUMOTO, Rae R et al.European journal of pharmacology. 2006, Vol 553, Num 1-3, pp 141-145, issn 0014-2999, 5 p.Article

Dextromethorphan attenuates trimethyltin-induced neurotoxicity via σ₁ receptor activation in ratsSHIN, Eun-Joo; NAH, Seung-Yeol; KIM, Hyoung-Chun et al.Neurochemistry international. 2007, Vol 50, Num 6, pp 791-799, issn 0197-0186, 9 p.Article

High affinity of sigma₁-binding sites for sterol isomerization inhibitors : evidence for a pharmacological relationship with the yeast sterol C₈-C₇ isomeraseMOEBIUS, F. F; REITER, R. J; HANNER, M et al.British journal of pharmacology. 1997, Vol 121, Num 1, pp 1-6, issn 0007-1188Article

Possible involvement of sigma-1 receptors in the anti-immobility action of bupropion, a dopamine reuptake inhibitorDHIR, Ashish; KULKARNI, S. K.Fundamental & clinical pharmacology. 2008, Vol 22, Num 4, pp 387-394, issn 0767-3981, 8 p.Article

Exploration of ring size in a series of cyclic vicinal diamines with σ₁ receptor affinityMOUSSA, Iman A; BANISTERA, Samuel D; MANOLI, Miral et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 17, pp 5493-5497, issn 0960-894X, 5 p.Article

Sigma-1 receptor-induced increase in murine spinal NR1 phosphorylation is mediated by the PKCα and ε, but not the PKCζ, isoformsROH, Dae-Hyun; YOON, Seo-Yeon; SEO, Hyoung-Sig et al.Neuroscience letters. 2010, Vol 477, Num 2, pp 95-99, issn 0304-3940, 5 p.Article

Inhibition of sigma-1 receptor reduces N-methyl-D-aspartate induced neuronal injury in methamphetamine-exposed and -naive hippocampiSMITH, Katherine J; BUTLER, Tracy R; PRENDERGAST, Mark A et al.Neuroscience letters. 2010, Vol 481, Num 3, pp 144-148, issn 0304-3940, 5 p.Article

A Mutation in Sigma-1 Receptor Causes Juvenile Amyotrophic Lateral SclerosisAL-SAIF, Amr; AL-MOHANNA, Futwan; BOHLEGA, Saeed et al.Annals of neurology. 2011, Vol 70, Num 6, pp 913-919, issn 0364-5134, 7 p.Article

Fluvoxamine as a sigma-1 receptor agonist improved cognitive impairments in a patient with schizophreniaIYO, Masaomi; SHIRAYAMA, Yukihiko; HASHIMOTO, Kenji et al.IYO, Masaomi; Progress in neuro-psychopharmacology & biological psychiatry. 2008, Vol 32, Num 4, pp 1072-1073, issn 0278-5846, 2 p.Article

Antitussive activity of sigma-1 receptor agonists in the guinea-pigBROWN, Claire; FEZOUI, Malika; SELIG, William M et al.British journal of pharmacology. 2004, Vol 141, Num 2, pp 233-240, issn 0007-1188, 8 p.Article

(+)-SKF-10,047 and dextromethorphan ameliorate conditioned fear stress through the activation of phenytoin-regulated σ₁ sitesKAMEI, H; KAMEYAMA, T; NABESHIMA, T et al.European journal of pharmacology. 1996, Vol 299, Num 1-3, pp 21-28, issn 0014-2999Article

Binding properties of SA4503, a novel and selective σ₁ receptor agonistMATSUNO, K; NAKAZAWA, M; OKAMOTO, K et al.European journal of pharmacology. 1996, Vol 306, Num 1-3, pp 271-280, issn 0014-2999, 9 p.Article

RLH-033, a novel, potent and selective ligand for the σ₁ recognition siteHUDKINS, R. L; MAILMAN, R. B; DEHAVEN-HUDKINS, D. L et al.European journal of pharmacology. 1994, Vol 271, Num 1, pp 235-236, issn 0014-2999Article

Straub tail reaction in mice treated with σ₁ receptor antagonist in combination with methamphetamineKITANAKA, Junichi; KITANAKA, Nobue; HALL, F. Scott et al.Brain research. 2012, Vol 1482, pp 40-46, issn 0006-8993, 7 p.Article

Sigma-1 receptor knockout mice display a depressive-like phenotypeSABINO, Valentina; COTTONE, Pietro; PARYLAK, Sarah L et al.Behavioural brain research. 2009, Vol 198, Num 2, pp 472-476, issn 0166-4328, 5 p.Article

Chronic treatment with a selective ligand for the sigma-1 receptor chaperone, SA4503, up-regulates BDNF protein levels in the rat hippocampusKIKUCHI-UTSUMI, Kazue; NAKAKI, Toshio.Neuroscience letters. 2008, Vol 440, Num 1, pp 19-22, issn 0304-3940, 4 p.Article

Understanding the molecular mechanism of sigma-1 receptors: Towards a hypothesis that sigma-1 receptors are intracellular amplifiers for signal transduction : Rational drug design and the discovery of the 1,2,3-triazolines as a unique class of anticonvulsants and antiischemic agentsSU, Tsung-Ping; HAYASHI, Teruo.Current medicinal chemistry. 2003, Vol 10, Num 20, pp 2073-2080, issn 0929-8673, 8 p.Article

Differences in cytochrome P450 forms involved in the metabolism of N, N-dipropyl-2-[4-methoxy-3-(2-phenylethoxy)phenyl]ethylamine monohydrochloride (NE-100), a novel sigma ligand, in human liver and intestineYAMAMOTO, Takahito; HAGIMA, Naoko; NAKAMURA, Masato et al.Drug metabolism and disposition. 2003, Vol 31, Num 1, pp 60-66, issn 0090-9556, 7 p.Article

Identification of a 27-kDa high affinity phenylalkylamine-binding polypeptide as the σ₁ binding site by photoaffinity labeling and ligand-directed antibodiesMOEBIUS, F. F; BURROWS, G. G; HANNER, M et al.Molecular pharmacology. 1993, Vol 44, Num 5, pp 966-971, issn 0026-895XArticle

Autoradiographic distribution of [³H](+)-pentazocine and [³H]1,3-di-o-tolylguanidine (DTG) binding sites in guinea pig brain : a comparative studyWALKER, J. M; BOWEN, W. D; GOLDSTEIN, S. R et al.Brain research. 1992, Vol 581, Num 1, pp 33-38, issn 0006-8993Article

Synthesis, σ₁, σ₂-receptors binding affinity and antiproliferative action of new C1-substituted adamantanesRIGANAS, Stefanos; PAPANASTASIOU, Ioannis; MOUTSOS, Vassilios I et al.Bioorganic & medicinal chemistry. 2012, Vol 20, Num 10, pp 3323-3331, issn 0968-0896, 9 p.Article

Sigma-1 ligands: Tic-hydantoin as a key pharmacophoreTOUSSAINT, Marion; MOUSSET, Deborah; FOULON, Catherine et al.European journal of medicinal chemistry. 2010, Vol 45, Num 1, pp 256-263, issn 0223-5234, 8 p.Article