1,2,4-Oxadiazoles: A new class of anti-prostate cancer agentsKHATIK, Gopal L; KAUR, Jasmine; KUMAR, Varun et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 5, pp 1912-1916, issn 0960-894X, 5 p.Article

2-Amidino analogs of glycine―amiloride conjugates: Inhibitors of urokinase-type plasminogen activatorMASSEY, Archna P; HARLEY, William R; PASUPULETI, Nagarekha et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 7, pp 2635-2639, issn 0960-894X, 5 p.Article

3-Phenyl-5-isothiazole carboxamides with potent mGluR1 antagonist activityFISHER, Matthew J; BACKER, Ryan T; LINGLIN LI et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 7, pp 2514-2517, issn 0960-894X, 4 p.Article

4-Piperidin-4-ylidenemethyl-benzamides as δ-opioid receptor agonists for CNS indications: Identifying clinical candidatesDANTZMAN, Cathy L; KING, Megan M; LIU, Jay et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 2, pp 1174-1178, issn 0960-894X, 5 p.Article

4-Substituted boro-proline dipeptides: Synthesis, characterization, and dipeptidyl peptidase IV, 8, and 9 activitiesWENGEN WU; YUXIN LIU; POPLAWSKI, Sarah E et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 17, pp 5536-5540, issn 0960-894X, 5 p.Article

4-Substituted-2-phenylquinazolines as inhibitors of BCRPJUVALE, Kapil; WIESE, Michael.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 21, pp 6766-6769, issn 0960-894X, 4 p.Article

5- and 6-Membered (thio)lactones are prodrug type carbonic anhydrase inhibitorsCARTA, Fabrizio; MARESCA, Alfonso; SCOZZAFAVA, Andrea et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 267-270, issn 0960-894X, 4 p.Article

A conformationally restricted uniconazole analogue as a specific inhibitor of rice ent-kaurene oxidase, CYP701A6TODOROKI, Yasushi; NAIKI, Kumi; MURAMATSU, Taku et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 9, pp 3240-3243, issn 0960-894X, 4 p.Article

A new class of pyrimidine nucleosides: inhibitors of hepatitis B and C virusesSHAKYA, Neeraj; VEDI, Satish; CHAO LIANG et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 20, pp 6475-6480, issn 0960-894X, 6 p.Article

A novel series of glucagon receptor antagonists with reduced molecular weight and lipophilicityFILIPSKI, Kevin J; JIANWEI BIAN; PERREAULT, Christian et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 415-420, issn 0960-894X, 6 p.Article

A specific molecular beacon probe for the detection of human prostate cancer cellsYU LIN JIANG; MCGOLDRICK, Christopher A; DELING YIN et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 11, pp 3632-3638, issn 0960-894X, 7 p.Article

A substituted 3,4-dihydropyrimidinone derivative (compound D22) prevents inflammation mediated neurotoxicity; role in microglial activation in BV-2 cellsOH WOOK KWON; MOON, Eunjung; CHARI, Murugulla A et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 16, pp 5199-5203, issn 0960-894X, 5 p.Article

A three-step protocol for lead optimization: Quick identification of key conformational features and functional groups in the SAR studies of non-ATP competitive MK2 (MAPKAPK2) inhibitorsXIANHAI HUANG; XIAOHONG ZHU; TRIVEDI, Prashant et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 65-70, issn 0960-894X, 6 p.Article

A β-tryptase inhibitor with a tropanylamide scaffold to improve in vitro stability and to lower hERG channel binding affinityGUYAN LIANG; CHOI-SLEDESKI, Yong Mi; JIESHENG KANG et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 4, pp 1606-1610, issn 0960-894X, 5 p.Article

Acremomannolipin A, the potential calcium signal modulator with a characteristic glycolipid structure from the filamentous fungus Acremonium strictumSUGIURA, Reiko; KITA, Ayako; TSUTSUI, Nozomi et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 21, pp 6735-6739, issn 0960-894X, 5 p.Article

Acyl derivatives of boswellic acids as inhibitors of NF-κB and STATsKUMAR, Ajay; SHAH, Bhahwal A; SINGH, Samar et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 431-435, issn 0960-894X, 5 p.Article

Acylprolinamides: A new class of peptide deformylase inhibitors with in vivo antibacterial activityAXTEN, Jeffrey M; MEDINA, Jesus R; KULKARNI, Swarupa et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 12, pp 4028-4032, issn 0960-894X, 5 p.Article

Amides of xanthurenic acid as zinc-dependent inhibitors of Lp-PLA₂LIN, Emme C. K; YI HU; ISHIYAMA, Junichi et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 2, pp 868-871, issn 0960-894X, 4 p.Article

Aminoimidazoles as BACE-1 inhibitors: The challenge to achieve in vivo brain efficacySWAHN, Britt-Marie; HOLENZ, Jörg; FÄLTING, Johanna et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 5, pp 1854-1859, issn 0960-894X, 6 p.Article

An improved microwave assisted one-pot synthesis, and biological investigations of some novel aryldiazenyl chromeno fused pyrrolidinesPARMAR, Narsidas J; PANSURIYA, Bhavesh R; BARAD, Hitesh A et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 12, pp 4075-4079, issn 0960-894X, 5 p.Article

Anion inhibition studies of an α-carbonic anhydrase from the thermophilic bacterium Sulfurihydrogenibium yellowstonense YO3AOP1DE LUCA, Viviana; VULLO, Daniela; SCOZZAFAVA, Andrea et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 17, pp 5630-5634, issn 0960-894X, 5 p.Article

Anti-inflammatory and PPAR trausaitivational effects of secondary metabolites from the roots of Asarum sieboldiiTRAN HONG QUANG; NGUYEN THI THANH NGAN; CHAU VAN MINH et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 7, pp 2527-2533, issn 0960-894X, 7 p.Article

Antibacterial activity of substituted dibenzo[a,g]quinolizin-7-ium derivativesPARHI, Ajit; SONGFENG LU; KELLEY, Cody et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 22, pp 6962-6966, issn 0960-894X, 5 p.Article

Anticonvulsant activity of artificial sweeteners: A structural link between sweet-taste receptor T1R3 and brain glutamate receptorsTALEVI, Alan; ENRIQUE, Andrea V; BRUNO-BLANCH, Luis E et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 12, pp 4072-4074, issn 0960-894X, 3 p.Article

Antimycobacterial activity: A facile three-component [3+2]-cycloaddition for the regioselective synthesis of highly functionalised dispiropyrrolidinesANG CHEE WEI; MOHAMED ASHRAF ALI; YEONG KENG YOON et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 15, pp 4930-4933, issn 0960-894X, 4 p.Article