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Results 1 to 25 of 680208

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STUDIES ON BIOLOGICALLY ACTIVE HALOGENATED COMPOUNDS. VI: SYNTHESIS AND ANTIBACTERIAL ACTIVITY OF FLUORINATED QUINOLINE DERIVATIVESTANI J; MUSHIKA Y; YAMAGUCHI T et al.1982; CHEM. PHARM. BULL.; ISSN 0009-2363; JPN; DA. 1982; VOL. 30; NO 10; PP. 3530-3543; BIBL. 12 REF.Article

STUDIES ON THE HETEROCYCLIC COMPOUNDS. XXI. A NEW ALKYLATION OF PYRIDAZINES WITH NITROMETHANE AND NITROETHANE.YANAI M; TAKEDA S; NISHIKAWA M et al.1977; CHEM. PHARM. BULL.; JAP.; DA. 1977; VOL. 25; NO 8; PP. 1856-1861; BIBL. 4 REF.Article

ACTION DE LA GUANIDINE ET DU THIOSEMICARBAZIDE SUR LES ESTERS OXALACETIQUES: OBTENTION DE DERIVES DE LA TRIAZINE-1,2,4 ET DU PYRAZOL PAR CYCLIZATION ALCALINEMAUDET D; GRANET R; PIEKARSKI S et al.1975; BULL. SOC. CHIM. FR.; FR.; DA. 1975; NO 11-12 PART. 2; PP. 2696-2702; ABS. ANGL.; BIBL. 17 REF.Article

ETUDE CHIMIQUE ET PHARMACOLOGIQUE D'UNE SERIE DE PYRIDAZONES SUBSTITUEESPITARCH L; CORONAS R; MALLOL J et al.1974; EUROP. J. MEDICIN. CHEM.; FR.; DA. 1974; VOL. 9; NO 6; PP. 644-650; ABS. ANGL. ALLEM.; BIBL. 33 REF.Article

NEW 4-PYRIDONYL-ACETAMIDO-CEPHALOSPORINS AND RELATED COMPOUNDSGERICKE P; ROGALSKI W.1979; ARZNEIMITTEL-FORSCH.; DEU; DA. 1979; VOL. 29; NO 2A; PP. 362-369; ABS. GER; BIBL. 7 REF.Article

4-DIALKYLAMINO-CHINOLINE UND 3,3-DISUBSTITUIERTE 4(3H)-CHINOLONE AUS 4H-3,1-BENZOXAZINONEN UND INAMINEN = DIALKYLAMINO-4 QUINOLEINES ET 3H-QUINOLONES-4 DISUBSTITUEES-3,3 A PARTIR DE 4H-BENZOOXAZINES-3,1 ET D'YNAMINESHOFLE G; HOLLITZER O; STEGLICH W et al.1972; ANGEW. CHEM.; DTSCH.; DA. 1972; VOL. 20; NO 15; PP. 716-718; BIBL. 9 REF.Serial Issue

SYNTHESIS AND ANTITRICHOMONAL ACTIVITY OF CERTAIN PYRAZOLO (1,5-A) PYRIMIDINESSENGA K; NOVINSON T; SPRINGER RH et al.1975; J. MEDICIN. CHEM.; U.S.A.; DA. 1975; VOL. 18; NO 3; PP. 312-314; BIBL. 15 REF.Article

SPECTROSCOPIC AND STRUCTURAL STUDIES OF QUINOLINE DERIVATIVES. II: FOURIER TRANSFORM I-R-SPECTROSCOPY. 1: ROTATIONAL ISOMERISM IN 3-ETHOXYCARBONYL-4 (1H)-QUINOLONE AND SOME OF ITS SUBSTITUTED DERIVATIVESMIREK J; URBANEK ZH.1981; SPECTROCHIM. ACTA, A; ISSN 0584-8539; GBR; DA. 1981; VOL. 37; NO 5; PP. 305-314; BIBL. 29 REF.Article

POTENTIAL WOOL GROWTH INHIBITORS. IMPROVED SYNTHESES OF MIMOSINE AND RELATED 4(1H)-PYRIDONES.HARRIS RLN.1976; AUSTRAL. J. CHEM.; AUSTRAL.; DA. 1976; VOL. 29; NO 6; PP. 1329-1334; BIBL. 18 REF.Article

THE GUERBET REACTION APPLIED TO DIODONEDINGJAN HA; CREZEE HA.1978; MIKROCHIM. ACTA; AUT; DA. 1978; VOL. 2; NO 5-6; PP. 395-402; ABS. GER; BIBL. 6 REF.Article

A convenient synthesis of 3-formyl-4(1H)-pyridonesARYA, F; BOUQUANT, J; CHUCHE, J et al.Synthesis (Stuttgart). 1983, Num 11, pp 946-948, issn 0039-7881Article

1-Ethyl-7-[3-[(ethylamino)methyl]-1-pyrrolidinyl]-6,8-difluoro-1,4-dihydro-4-oxo-3-quinoline-carboxylic acid. New quinolone antibacterial with potent gram-positive activityDOMAGALA, J. M; HEIFETZ, C. L; MICH, T. F et al.Journal of medicinal chemistry (Print). 1986, Vol 29, Num 4, pp 445-448, issn 0022-2623Article

SYNTHESE EINIGER 4-OXO-3.4-DIHYDROCHINAZOLIN-3-CARBONSAEURE-DERIVATE. = SYNTHESE DE QUELQUES DERIVES DE L'ACIDE OXO-4 DIHYDRO-3,4 QUINAZOLINE CARBOXYLIQUE-3JOHNE S; JUNG B.1978; PHARMAZIE; DDR; DA. 1978; VOL. 33; NO 5; PP. 298-299; BIBL. 9 REF.Article

Mass spectroscopy of natural products. XX: Quinazoline carboxylic acids. IV: Comparative positive and negative ion mass spectroscopic studies of 3,4-dihydroquinazolin-4-on-3-ylalkanoic acids and 3,4-dihydro-1,2,3-benzotriazin-4-on-3-ylalkanoic acidsSCHMIDT, J; SÜSSE, M; JOHNE, S et al.Organic mass spectrometry. 1985, Vol 20, Num 3, pp 184-188, issn 0030-493XArticle

Novel amino-substituted 3-quinolinecarboxylic acid antibacterial agents: synthesis and structure-activity relationshipsWENTLAND, M. P; BAILEY, D. M; CORNETT, J. B et al.Journal of medicinal chemistry (Print). 1984, Vol 27, Num 9, pp 1103-1108, issn 0022-2623Article

ETUDES DANS LE DOMAINE DES LACTONES NON SATUREES. XXIII. SYNTHESE DES ETHOXYCARBONYL-4 BROMO-5 TRIALKYL-5,6,6 DIHYDRO-5,6 PYRONES-2AVETISYAN AA; AKOPYAN KG; DANGYAN MT et al.1974; ARM. KHIM. ZH.; S.S.S.R.; DA. 1974; VOL. 27; NO 5; PP. 408-410; ABS. ARM. ANGL.; BIBL. 3 REF.Article

Nitrogen bridgehead compounds. LI: Autoxidation of 9-aminotetrahydro-4H-pyrido[1,2-a]pyrimidin-4-ones. Synthesis and stereochemistry of 9-amino- and 9-hydroxy-6,7-dihydro-4H-pyrido[1,2-a]-pyrimidin-4-onesBREINING, T; HERMECZ, I; PODANYI, B et al.Journal of heterocyclic chemistry. 1985, Vol 22, Num 5, pp 1253-1259, issn 0022-152XArticle

Synthesis of substituted 9-oxo-9,10-dihydro-acridine-4-carboxyclic acids. I: Factors affecting the direction of ring closure of substituted N-(2-carboxyphenylamino)benzoic acidsSTEWART, G. M; REWCASTLE, G. W; DENNY, W. A et al.Australian journal of chemistry. 1984, Vol 37, Num 9, pp 1939-1950, issn 0004-9425Article

Synthesis and antimicrobial evaluation of a series of 7-[3-amino (or aminomethyl)-4-aryl (or cyclopropyl)-1-pyrrolidinyl]-4-quinolone- and -1,8-naphthyridone-3-carboxylic acidsBUCSH, R. A; DOMAGALA, J. M; LABORDE, E et al.Journal of medicinal chemistry (Print). 1993, Vol 36, Num 26, pp 4139-4151, issn 0022-2623Article

Action of the benzodiazepine antagonist Ro 15-1788 in humans after sleep withdrawalEMRICH, H. M; SONDEREGGER, P; MAI, N et al.Neuroscience letters. 1984, Vol 47, Num 3, pp 369-373, issn 0304-3940Article

UNTERSUCHUNGEN UEBER DIE ANTIBAKTERIELLE AKTIVITAET VON CHINOLONCARBONSAEUREN. IX. AZAANALOGA. DI- UND TRISUBSTITUIERTE 1,4-DIHYDRO-4-OXO-1,5-NAPHTHYRIDIN-3-CARBONSAEUREN UND 1-AETHYL-4-PYRIDON-3-CARBONSAEURE. = RECHERCHES SUR L'ACTIVITE ANTIBACTERIENNE DES ACIDES QUINOLONECARBOXYLIQUES. IX. AZAANALOGUES. ACIDES DIHYDRO-1,4 OXO-4 NAPHTYRIDINE-1,5 CARBOXYLIQUES-3 DI- ET TRISUBSTITUES ET ACIDE ETHYL-1 PYRIDONE-4 CARBOXYLIQUE-3HEINDL J; KELM HW; DOGS E et al.1977; EUROP. J. MEDICIN. CHEM.; FR.; DA. 1977; VOL. 12; NO 6; PP. 549-555; ABS. ANGL. FR.; BIBL. 22 REF.Article

2,5-DICARBONYL SUGARS: NEW INTERMEDIATES FOR SYNTHESISING HETEROCYCLIC RINGS. I. SYNTHESIS OF 4(LH)-PYRIDAZINONE DERIVATIVES FROM DICARBONYL SUGARSIMADA K; ASANO K.1974; CHEM. PHARM. BULL.; JAP.; DA. 1974; VOL. 22; NO 8; PP. 1691-1698; BIBL. 14 REF.Article

ACIDES ALKYL-1-OXO-4-DIHYDRO-1.4 PYRIDO (2.3-B) QUINOXALINE-3 CARBOXYLIQUES A ACTION ANTIBACTERIENNEPESSON M; DE LAJUDIE P; ANTOINE M et al.1976; C.R. ACAD. SCI., C; FR.; DA. 1976; VOL. 282; NO 17; PP. 861-864; ABS. ANGL.; BIBL. 10 REF.Article

EXISTENCE OF ALTERNATIVE TAUTOMERS OF HETEROCYCLIC HYDRAZINE DERIVATIVES IN THE CRYSTALLINE STATELE COUNT DJ; GREER AT.1973; TETRAHEDRON LETTERS; G.B.; DA. 1973; NO 31; PP. 2905-2906; BIBL. 3 REF.Serial Issue

GENERAL SYNTHESIS OF: 5-SUBSTITUTED-3-ACYL-4-CARBETHOXYPYRAZOLES, 3,6-SUBSTITUTED-5-CARBETHOXY-4 (1H) PYRIDAZINONES AND 3,7-SUBSTITUTED-PYRAZOLO (3,4-D) PYRIDAZINE-4 (5H) ONES VIA REACTIONS BETWEEN 2-HYDROXY, METHOXY, AND ACETOXY-3 (2H) FURANONES AND HYDRAZINE.GELIN S; GELIN R.1977; J. HETEROCYCL. CHEM.; U.S.A.; DA. 1977; VOL. 14; NO 1; PP. 75-79; BIBL. 17 REF.Article

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