4-[1-(Substituted aryl/alkyl carbonyl)-benzoimidazol-2-yl]-benzenesulfonic acids: Synthesis, antimicrobial activity, QSAR studies, and antiviral evaluation
- Auteur
- YADAV, Snehlata1 ; KUMAR, Pradeep1 ; DE CLERCQ, Erik2 ; BALZARINI, Jan2 ; PANNECOUQUE, Christophe2 ; SHARWAN KUMAR DEWAN3 ; NARASIMHAN, Balasubramanian1
[1] Faculty of Pharmaceutical Sciences, Maharshi Dayanand University, Rohtak 124001, India
[2] Laboratory of Virology & Chemotherapie, Rega Institute for Medical Research, Minderbroedersstraat 10, 3000 Leuven, Belgium
[3] Department of Chemistry, Maharshi Dayanand University, Rohtak 124001, India - Source
European journal of medicinal chemistry. 2010, Vol 45, Num 12, pp 5985-5997, 13 p ; ref : 51 ref
- CODEN
- EJMCA5
- ISSN
- 0223-5234
- Domaine scientifique
- Organic chemistry; Pharmacology drugs
- Editeur
- Elsevier, Kidlington
- Pays de publication
- United Kingdom
- Type de document
- Article
- Langue
- English
- Mot clé auteur
- Antimicrobial Antiviral Benzimidazoles QSAR
- Mot clé (fr)
- Acide sulfonique Antibactérien Antifongique Antimicrobien Antiviral Carboxamide Composé aliphatique Composé aromatique Composé bicyclique Dérivé du benzimidazole Dérivé du benzène Hétérocycle azote In vitro Prédiction Relation structure activité Synthèse chimique Benzènesulfonique acide(4-[1-(4-nitrobenzoyl)benzimidazol-2-yl]) Benzènesulfonique acide(4-[1-octadéc-9-énoylbenzimidazol-2-yl]) QSAR
- Mot clé (en)
- Sulfonic acid Antibacterial agent Antifungal agent Antimicrobial agent Antiviral Carboxamide Aliphatic compound Aromatic compound Bicyclic compound Benzimidazole derivatives Benzene derivatives Nitrogen heterocycle In vitro Prediction Structure activity relation Chemical synthesis
- Mot clé (es)
- Acido sulfónico Antibacteriano Antifúngico Antimicrobiano Antiviral Carboxamida Compuesto alifático Compuesto aromático Compuesto bicíclico Benzimidazol derivado Benceno derivado Heterociclo nitrógeno In vitro Predicción Relación estructura actividad Síntesis química
- Classification
- Pascal
- 002 Sciences biologiques et medicales / 002B Sciences medicales / 002B02 Pharmacologie. Traitements medicamenteux / 002B02S Antibiotiques. Antiinfectieux. Antiparasitaires / 002B02S01 Généralités
- Pascal
- 002 Sciences biologiques et medicales / 002B Sciences medicales / 002B02 Pharmacologie. Traitements medicamenteux / 002B02S Antibiotiques. Antiinfectieux. Antiparasitaires / 002B02S02 Antibactériens
- Pascal
- 002 Sciences biologiques et medicales / 002B Sciences medicales / 002B02 Pharmacologie. Traitements medicamenteux / 002B02S Antibiotiques. Antiinfectieux. Antiparasitaires / 002B02S04 Antifongiques
- Pascal
- 002 Sciences biologiques et medicales / 002B Sciences medicales / 002B02 Pharmacologie. Traitements medicamenteux / 002B02S Antibiotiques. Antiinfectieux. Antiparasitaires / 002B02S05 Antiviraux
- Discipline
- Pharmacological treatments
- Provenance
- Inist-CNRS
- Base de données
- PASCAL
- Identifiant INIST
- 23474192
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.ejmech.2010.09.065 
https://dx.doi.org/10.1016/j.ejmech.2010.09.065
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