Design and synthesis of 3-(azol-1-yl)phenylpropanes as microbicidal spermicides for prophylactic contraception
- Auteur
- KUMAR, Lalit1 ; SARSWAT, Amit1 ; SHARMA, Vishnu L1 ; LAL, Nand1 ; JAIN, Ashish2 ; KUMAR, Sumit3 ; KIRAN KUMAR, S. T. V. S1 ; MAIKHURI, Jagdamba P2 ; PANDEY, Atindra K4 ; SHUKLA, Praveen K4 ; GUPTA, Gopal2
[1] Division of Medicinal and Process Chemistry, Central Drug Research Institute (CSIR), Lucknow 226 001, India
[2] Division of Endocrinology, Central Drug Research Institute (CSIR), Lucknow 226 001, India
[3] National Institute of Pharmaceutical Education and Research (NIPER), Raebareli 229 010, India
[4] Division of Fermentation Technology, Central Drug Research Institute (CSIR), Lucknow 226 001, India - Source
Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 1, pp 176-181, 6 p
- ISSN
- 0960-894X
- Domaine scientifique
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Editeur
- Elsevier, Amsterdam
- Pays de publication
- Netherlands
- Type de document
- Article
- Langue
- English
- Mot clé auteur
- Anticandida Antitrichomonas Fluoxetine Nonoxynol-9 Spermicides
- Mot clé (fr)
- Activité biologique Antifongique Antimicrobien Antiparasitaire Antiprotozoaire Candida Compatibilité Contraceptif Cétone Dérivé d'azole Dérivé du benzimidazole Fluoxétine Lactobacillus Neurotransmetteur Spermicide Synthèse chimique Trichomonas vaginalis Benzimidazole(1-[2-benzoyléthyl]) Imidazole(1-[2-benzoyléthyl]-4-nitro) Bactérie Fungi Imperfecti Fungi Inhibiteur recapture Lactobacillaceae Protozoa Sérotonine Trichomonadida
- Mot clé (en)
- Biological activity Antifungal agent Antimicrobial agent Parasiticide Antiprotozoal agent Candida Compatibility Contraceptive Ketone Azole derivatives Benzimidazole derivatives Fluoxetine Lactobacillus Neurotransmitter Spermicide Chemical synthesis Trichomonas vaginalis Bacteria Fungi Imperfecti Fungi Reuptake inhibitor Lactobacillaceae Protozoa Serotonin Trichomonadida
- Mot clé (es)
- Actividad biológica Antifúngico Antimicrobiano Antiparasitario Antiprotozoario Candida Compatibilidad Anticonceptivo Cetona Azol derivado Benzimidazol derivado Fluoxetina Lactobacillus Neurotransmisor Espermicida Síntesis química Trichomonas vaginalis Bacteria Fungi Imperfecti Fungi Inhibidor recaptura Lactobacillaceae Protozoa Serotonina Trichomonadida
- Classification
- Pascal
- 002 Sciences biologiques et medicales / 002B Sciences medicales / 002B02 Pharmacologie. Traitements medicamenteux / 002B02P Appareil génital. Reproduction
- Pascal
- 002 Sciences biologiques et medicales / 002B Sciences medicales / 002B02 Pharmacologie. Traitements medicamenteux / 002B02S Antibiotiques. Antiinfectieux. Antiparasitaires / 002B02S01 Généralités
- Pascal
- 002 Sciences biologiques et medicales / 002B Sciences medicales / 002B02 Pharmacologie. Traitements medicamenteux / 002B02S Antibiotiques. Antiinfectieux. Antiparasitaires / 002B02S04 Antifongiques
- Pascal
- 002 Sciences biologiques et medicales / 002B Sciences medicales / 002B02 Pharmacologie. Traitements medicamenteux / 002B02S Antibiotiques. Antiinfectieux. Antiparasitaires / 002B02S06 Antiparasitaires
- Discipline
- Pharmacological treatments
- Provenance
- Inist-CNRS
- Base de données
- PASCAL
- Identifiant INIST
- 23726777
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2010.11.042 
https://dx.doi.org/10.1016/j.bmcl.2010.11.042
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