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Discovery of a series of potent and selective human H4 antagonists using ligand efficiency and libraries to explore structure-activity relationship (SAR)ABID MASOOD, M; SELBY, Matthew D; LIU, Wai L et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 21, pp 6591-6595, issn 0960-894X, 5 p.Article

Computational screening for membrane-directed inhibitors of mast cell activationBATISTA, José; FRIEDRICHSON, Tim; SCHLECHTINGEN, Georg et al.European journal of medicinal chemistry. 2010, Vol 45, Num 6, pp 2700-2704, issn 0223-5234, 5 p.Article

Exploration of SAR features by modifications of thiazoleacetic acids as CRTH2 antagonistsGRIMSTRUP, Marie; RECEVEUR, Jean-Marie; RIST, Oystein et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 5, pp 1638-1641, issn 0960-894X, 4 p.Article

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Core exploration in optimization of chemokine receptor CCR4 antagonistsPURANDARE, Ashok V; HONGHE WAN; SOMERVILLE, John E et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 3, pp 679-682, issn 0960-894X, 4 p.Article

4-Acyl-1-(4-aminoalkoxyphenyl)-2-ketopiperazines as a Novel Class of Non-Brain-Penetrant Histamine H₃ Receptor AntagonistsPROCOPIOU, Panayiotis A; ANCLIFF, Rachael A; MORRISS, Karen M. L et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 26, pp 6706-6717, issn 0022-2623, 12 p.Article

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Small molecule inhibitors of IgE synthesisBROWN, Alan; HENDERSON, Alan; LANE, Charlotte et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 17, pp 4697-4699, issn 0960-894X, 3 p.Article

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Effect of probiotic Lactobacillus strains in children with atopic dermatitisROSENFELDT, Vibeke; BENFELDT, Eva; DAM NIELSEN, Susanne et al.Journal of allergy and clinical immunology. 2003, Vol 111, Num 2, pp 389-395, issn 0091-6749, 7 p.Article

In vitro inhibition of human conjunctival mast-cell degranulation by ketotifenSCHOCH, C.Journal of ocular pharmacology and therapeutics. 2003, Vol 19, Num 1, pp 75-81, issn 1080-7683, 7 p.Article

Inhibition of histamine H₁ receptor downregulation by KT5823, a protein kinase g inhibitorMIYOSHI, K; KAWAKAMI, N; HORIO, S et al.Methods and findings in experimental and clinical pharmacology. 2003, Vol 25, Num 5, pp 343-347, issn 0379-0355, 5 p.Article

Inhibitory effects of ketotifen on eotaxin-dependent activation of eosinophils: consequences for allergic eye diseasesWOERLY, G; LOISEAU, S; LOYENS, M et al.Allergy (Copenhagen). 2003, Vol 58, Num 5, pp 397-406, issn 0105-4538, 10 p.Article

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Pharmacotherapy for allergic rhinitis: a critical review of leukotriene receptor antagonists compared with other treatmentsNATHAN, Robert A.Annals of allergy, asthma, & immunology. 2003, Vol 90, Num 2, pp 182-191, issn 1081-1206, 10 p.Article